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Digest: Richard A. Glennon: literature collection | Please login to post | |
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Lego (Hive Bee) 10-25-04 15:00 No 506957 
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Richard A. Glennon: literature collection (Rated as: excellent) |
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The literature was collected with a PubMed search and with the collection on Glennon's Homepage. All fulltexts available either at the Hive or at Rhodium's page will be hyperlinked. Suggestions are welcome! Thanks to 7is, Nicodem and Rhodium for providing scanned articles!  Please report dead links either at Post 506981 (Aurelius: "Glennon Digest", General Discourse) or via PM. Version 1.00: All PubMed entries and articles from Glennon's homepage are collected (new entries compared to the beta version can bee found by the right format) Version 1.01: All articles were sorted in different chapters, all articles of interest from J. Med. Chem. were uploaded Version 1.10: All articles retrieved by 7is were uploaded, all entries now have a proper format  Richard A. Glennon's Homepage (http://www.phc.vcu.edu/Faculty/Glennon.html) 5-HT2A/C ligands and other hallucinogens: synthesis and pharmacology Glennon RA, Bondarev ML, Khorana N, Young R, May JA, Hellberg MR, McLaughlin MA, Sharif NA beta-Oxygenated Analogues of the 5-HT2A Serotonin Receptor Agonist 1-(4-Bromo-2,5-dimethoxyphenyl)-2-aminopropane J. Med. Chem., 2004, DOI:10.1021/jm040082s Post 537524 (Lego: "Glennon: Oxygenated DOB analogues", Novel Discourse)  Peddi S, Roth BL, Glennon RA, Westkaemper RB Structural determinants for high 5-HT2A receptor affinity of spiro[9,10-dihydroanthracene]-9,3(')-pyrrolidine (SpAMDA) Bioorg. Med. Chem. Lett., 2004, 14(9), 2279-2283 Medline (PMID=15081025) Peddi S, Roth BL, Glennon RA, Westkaemper RB Spiro[9,10-dihydroanthracene]-9,3'-pyrrolidine-a structurally unique tetracyclic 5-HT2A receptor antagonist Eur. J. Pharmacol., 2003, 482(1-3), 335-337 Medline (PMID=14660041) Grella B, Teitler M, Smith C, Herrick-Davis K, Glennon RA Binding of beta-carbolines at 5-HT2 serotonin receptors Bioorg. Med. Chem. Lett., 2003, 13(24), 4421-4425 Medline (PMID=14643338) Post 506956 (Lego: "Binding of beta-carbolines at 5-HT2 receptors", General Discourse) Eckler JR, Chang-Fong J, Rabin RA, Smith C, Teitler M, Glennon RA, Winter JC Behavioral characterization of 2-O-desmethyl and 5-O-desmethyl metabolites of the phenylethylamine hallucinogen DOM Pharmacol. Biochem. Behav., 2003, 75(4), 845-852 Medline (PMID=12957227) Post 474567 (Rhodium: "Recent Psychedelic Pharmacology Research", General Discourse) Peddi S, Roth BL, Glennon RA, Westkaemper RB Ring substituted analogues of 5-aminomethyl-10,11-dihydro-dibenzo[a,d]cycloheptene (AMDH): potential modes of binding to the 5-HT2A receptor Bioorg. Med. Chem. Lett., 2003, 13(15), 2565-2568 Medline (PMID=12852967) Westkaemper RB, Glennon RA Application of ligand SAR, receptor modeling and receptor mutagenesis to the discovery and development of a new class of 5-HT2A ligands Curr. Top. Med. Chem., 2002, 2(6), 575-598 Medline (PMID=12052195) Post 504089 (Lego: "Glennon on SAR and new 5-HT2A ligands", Novel Discourse) Glennon RA, Metwally K, Dukat M, Ismaiel AM, De los Angeles J, Herndon J, Teitler M, Khorana N Ketanserin and spiperone as templates for novel serotonin 5-HT2A antagonists Curr. Top. Med. Chem., 2002, 2(6), 539-558 Medline (PMID=12052193) Chang-Fong J, Addo J, Dukat M, Smith C, Mitchell NA, Herrick-Davis K, Teitler M, Glennon RA Evaluation of isotryptamine derivatives at 5-HT2 serotonin receptors Bioorg. Med. Chem. Lett., 2002, 12(2), 155-158 Medline (PMID=11755343) Rangisetty JB, Dukat M, Dowd CS, Herrick-Davis K, DuPre A, Gadepalli S, Teitler M, Kelley CR, Sharif NA, Glennon RA 1-[2-methoxy-5-(3-phenylpropyl)]-2-aminopropane unexpectedly shows 5-HT2A serotonin receptor affinity and antagonist character J. Med. Chem., 2001, 44(20), 3283-3291 Medline (PMID=11563927) Dowd CS, Herrick-Davis K, Egan C, DuPre A, Smith C, Teitler M, Glennon RA 1-[4-(3-Phenylalkyl)phenyl]-2-aminopropanes as 5-HT2A partial agonists J. Med. Chem., 2000, 43(16), 3074-3084 Medline (PMID=10956215) https://www.rhodium.ws/pdf/glennon.partial.agonists.pdf Glennon RA, Dukat M, Grella B, Hong S, Costantino L, Teitler M, Smith C, Egan C, Davis K, Mattson MV Binding of beta-carbolines and related agents at serotonin (5-HT2 and 5-HT1A), dopamine (D2) and benzodiazepine receptors Drug Alcohol Depend., 2000, 60(2), 121-132 Medline (PMID=10940539) Post 494854 (Nicodem: "Papers on beta-carbolines", General Discourse) Kristiansen K, Kroeze WK, Willins DL, Gelber EI, Savage JE, Glennon RA, Roth BL A highly conserved aspartic acid (Asp-155) anchors the terminal amine moiety of tryptamines and is involved in membrane targeting of the 5-HT2A serotonin receptor but does not participate in activation via a "salt-bridge disruption" mechanism J. Pharmacol. Exp. Ther., 2000, 293(3), 735-746 Medline (PMID=10869371) Westkaemper RB, Runyon SP, Bondarev ML, Savage JE, Roth BL, Glennon RA 9-(Aminomethyl)-9,10-dihydroanthracene is a novel and unlikely 5-HT2A receptor antagonist Eur. J. Pharmacol., 1999, 380(1), R5-7 Medline (PMID=10513561) Nelson DL, Lucaites VL, Wainscott DB, Glennon RA Comparisons of hallucinogenic phenylisopropylamine binding affinities at cloned human 5-HT2A, 5-HT2B and 5-HT2C receptors Naunyn Schmiedebergs Arch. Pharmacol., 1999, 359(1), 1-6 Medline (PMID=9933142) Metwally KA, Dukat M, Egan CT, Smith C, DuPre A, Gauthier CB, Herrick-Davis K, Teitler M, Glennon RA Spiperone: influence of spiro ring substituents on 5-HT2A serotonin receptor binding J. Med. Chem., 1998, 41(25), 5084-5093 Medline (PMID=9836624) Egan CT, Herrick-Davis K, Miller K, Glennon RA, Teitler M Agonist activity of LSD and lisuride at cloned 5HT2A and 5HT2C receptors Psychopharm. (Berl)., 1998, 136(4), 409-414 Medline (PMID=9600588) Ismaiel AM, Arruda K, Teitler M, Glennon RA Ketanserin analogues: the effect of structural modification on 5-HT2 serotonin receptor binding J. Med. Chem., 1995, 38(7), 1196-1202 Medline (PMID=7707322) Choudhary MS, Sachs N, Uluer A, Glennon RA, Westkaemper RB, Roth BL Differential ergoline and ergopeptine binding to 5-hydroxytryptamine2A receptors: ergolines require an aromatic residue at position 340 for high affinity binding Mol. Pharmacol., 1995, 47(3), 450-457 Medline (PMID=7700242) Glennon RA, Dukat M, el-Bermawy M, Law H, De los Angeles J, Teitler M, King A, Herrick-Davis K Influence of amine substituents on 5-HT2A versus 5-HT2C binding of phenylalkyl- and indolylalkylamines J. Med. Chem., 1994, 37(13), 1929-1935 Medline (PMID=8027974) Post 495672 (scarmani: "N-(4-Bromobenzyl)-5-methoxytryptamine Bioassay", General Discourse) Westkaemper RB, Glennon RA Molecular modeling of the interaction of LSD and other hallucinogens with 5-HT2 receptors NIDA Res Monogr., 1994, 146, 263-283 Medline (PMID=8742803) Ismaiel AM, De Los Angeles J, Teitler M, Ingher S, Glennon RA Antagonism of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane stimulus with a newly identified 5-HT2- versus 5-HT1C-selective antagonist J. Med. Chem., 1993, 36(17), 2519-2525 Medline (PMID=8355253) Herndon JL, Ismaiel A, Ingher SP, Teitler M, Glennon RA Ketanserin analogues: structure-affinity relationships for 5-HT2 and 5-HT1C serotonin receptor binding J. Med. Chem., 1992, 35(26), 4903-4910 Medline (PMID=1479590) Darmani NA, Martin BR, Glennon RA Repeated administration of low doses of cocaine enhances the sensitivity of 5-HT2 receptor function Pharmacol. Biochem. Behav., 1992, 41(3), 519-527 Medline (PMID=1584831) Post 512438 (7is: "All the missing PBB articles part 1", General Discourse) Glennon RA, Raghupathi R, Bartyzel P, Teitler M, Leonhardt S Binding of phenylalkylamine derivatives at 5-HT1C and 5-HT2 serotonin receptors: evidence for a lack of selectivity J. Med. Chem., 1992, 35(4), 734-740 Medline (PMID=1542100) http://nic-nac-project.de/~tajkor/jm00082a014.pdf Darmani NA, Martin BR, Pandey U, Glennon RA Inhibition of 5-HT2 receptor-mediated head-twitch response by cocaine via indirect stimulation of adrenergic alpha 2 and serotonergic 5-HT1A receptors Pharmacol. Biochem. Behav., 1991, 38(2), 353-367 Medline (PMID=1676173) Post 512438 (7is: "All the missing PBB articles part 1", General Discourse) Appel NM, Mitchell WM, Garlick RK, Glennon RA, Teitler M, De Souza EB Autoradiographic characterization of (+-)-1-(2,5-dimethoxy-4-[125I] iodophenyl)-2-aminopropane ([125I]DOI) binding to 5-HT2 and 5-HT1c receptors in rat brain J. Pharmacol. Exp. Ther., 1990, 255(2), 843-857 Medline (PMID=2243353) Glennon RA, Chaurasia C, Titeler M Binding of indolylalkylamines at 5-HT2 serotonin receptors: examination of a hydrophobic binding region J. Med. Chem., 1990, 33(10), 2777-2784 Medline (PMID=2213830) Glennon RA Do classical hallucinogens act as 5-HT2 agonists or antagonists? Neuropsychopharmacology, 1990, 3(5-6), 509-517 Medline (PMID=2078284) Darmani NA, Martin BR, Glennon RA Withdrawal from chronic treatment with (+/-)-DOI causes super-sensitivity to 5-HT2 receptor-induced head-twitch behaviour in mice Eur. J. Pharmacol., 1990, 186(1), 115-118 Medline (PMID=2282932) Darmani NA, Martin BR, Pandey U, Glennon RA Do functional relationships exist between 5-HT1A and 5-HT2 receptors? Pharmacol. Biochem. Behav., 1990, 36(4), 901-906 Medline (PMID=2145593) Post 512438 (7is: "All the missing PBB articles part 1", General Discourse) Seggel MR, Yousif MY, Lyon RA, Titeler M, Roth BL, Suba EA, Glennon RA A structure-affinity study of the binding of 4-substituted analogues of 1-(2,5-dimethoxyphenyl)-2-aminopropane at 5-HT2 serotonin receptors J. Med. Chem., 1990, 33(3), 1032-1036 Medline (PMID=2308135) https://www.rhodium.ws/pdf/glennon.sar.4-subst.pea.pdf Sadzot B, Baraban JM, Glennon RA, Lyon RA, Leonhardt S, Jan CR, Titeler M Hallucinogenic drug interactions at human brain 5-HT2 receptors: implications for treating LSD-induced hallucinogenesis Psychopharm. (Berl)., 1989, 98(4), 495-499 Medline (PMID=2505289) Lyon RA, Titeler M, Seggel MR, Glennon RA Indolealkylamine analogs share 5-HT2 binding characteristics with phenylalkylamine hallucinogens Eur. J. Pharmacol., 1988, 145(3), 291-297 Medline (PMID=3350047) Glennon RA, Seggel MR, Soine WH, Herrick-Davis K, Lyon RA, Titeler M [125I]-1-(2,5-dimethoxy-4-iodophenyl)-2-amino-propane: an iodinated radioligand that specifically labels the agonist high-affinity state of 5-HT2 serotonin receptors J. Med. Chem., 1988, 31(1), 5-7 Medline (PMID=3336031) https://www.rhodium.ws/pdf/glennon.doi-125.pdf Titeler M, Lyon RA, Glennon RA Radioligand binding evidence implicates the brain 5-HT2 receptor as a site of action for LSD and phenylisopropylamine hallucinogens Psychopharm. (Berl)., 1988, 94(2), 213-216 Medline (PMID=3127847) Titeler M, Lyon RA, Davis KH, Glennon RA Selectivity of serotonergic drugs for multiple brain serotonin receptors. Role of [3H]-4-bromo-2,5-dimethoxyphenylisopropylamine ([3H]DOB), a 5-HT2 agonist radioligand Biochem Pharmacol., 1987, 36(19), 3265-3271 Medline (PMID=3663239) Seggel MR, Qureshi GD, Glennon RA Effect of 5-HT2-selective agonists on cat platelet aggregation Life Sci., 1987, 41(9), 1077-1081 Medline (PMID=3613863) Post 508288 (7is: "All the missing Life Sciences articles part 2", General Discourse) Glennon RA, Titeler M, Seggel MR, Lyon RA N-methyl derivatives of the 5-HT2 agonist 1-(4-bromo-2,5-dimethoxyphenyl)-2-aminopropane J. Med. Chem., 1987, 30(5), 930-932 Medline (PMID=3572981) Rasmussen K, Glennon RA, Aghajanian GK Phenethylamine hallucinogens in the locus coeruleus: potency of action correlates with rank order of 5-HT2 binding affinity Eur. J. Pharmacol., 1986, 132(1), 79-82 Medline (PMID=3816969) Glennon RA, Slusher RM, Lyon RA, Titeler M, McKenney JD 5-HT1 and 5-HT2 binding characteristics of some quipazine analogues J. Med. Chem., 1986, 29(11), 2375-2380 Medline (PMID=3783595) Young R, Rosecrans JA, Glennon RA Further studies on the dose-dependent stimulus properties of 5-methoxy-N,N-dimethyltryptamine Pharmacol. Biochem. Behav., 1986 , 25(6), 1207-1210 Medline (PMID=3809222) Post 512438 (7is: "All the missing PBB articles part 1", General Discourse) Glennon RA Discriminative stimulus properties of the serotonergic agent 1-(2,5-dimethoxy-4-iodophenyl)-2-aminopropane (DOI) Life Sci., 1986, 39(9), 825-830 Medline (PMID=2943960) Post 508288 (7is: "All the missing Life Sciences articles part 2", General Discourse) Glennon RA Discriminative stimulus properties of the 5-HT1A agonist 8-hydroxy-2-(di-n-propylamino)tetralin (8-OH DPAT) Pharmacol. Biochem. Behav., 1986, 25(1), 135-139 Medline (PMID=2944129) Post 512438 (7is: "All the missing PBB articles part 1", General Discourse) Glennon RA Discriminative stimulus properties of phenylisopropylamine derivatives Drug Alcohol Depend., 1986, 17(2-3), 119-134 Medline (PMID=2874967) Glennon RA, McKenney JD, Lyon RA, Titeler M 5-HT1 and 5-HT2 binding characteristics of 1-(2,5-dimethoxy-4-bromophenyl)-2-aminopropane analogues J. Med. Chem., 1986, 29(1), 194-199 Medline (PMID=3950904) Glennon RA, Titeler M, Young R Structure-activity relationships and mechanism of action of hallucinogenic agents based on drug discrimination and radioligand binding studies Psychopharmacol Bull., 1986, 22(3), 953-958 Medline (PMID=3025916) Glennon RA, Hauck AE Mechanistic studies on DOM as a discriminative stimulus Pharmacol. Biochem. Behav., 1985, 23(6), 937-941 Medline (PMID=2934750) Post 512438 (7is: "All the missing PBB articles part 1", General Discourse) Glennon RA, Young R, Hauck AE Structure-activity studies on methoxy-substituted phenylisopropylamines using drug discrimination methodology Pharmacol. Biochem. Behav., 1985, 22(5), 723-729 Medline (PMID=3839309) Post 512438 (7is: "All the missing PBB articles part 1", General Discourse) Glennon RA, Titeler M, McKenney JD Evidence for 5-HT2 involvement in the mechanism of action of hallucinogenic agents Life Sci., 1984, 35(25), 2505-2511 Medline (PMID=6513725) Post 508287 (not existing) Glennon RA, Jacyno JM, Young R, McKenney JD, Nelson D Synthesis and evaluation of a novel series of N,N-dimethylisotryptamines J. Med. Chem., 1984, 27(1), 41-45 Medline (PMID=6581313) Glennon RA, Jacyno JM, Young R A comparison of the behavioral properties of (±)-, (-)-, and (+)-5-methoxy-alpha-methyltryptamine Biol. Psychiatry., 1983, 18(4), 493-498 Medline (PMID=6860723) Glennon RA, Young R, Jacyno JM Indolealkylamine and phenalkylamine hallucinogens. Effect of alpha-methyl and N-methyl substituents on behavioral activity Biochem Pharmacol. 1983, 32(7), 1267-1273 Medline (PMID=6573879) https://www.rhodium.ws/pdf/butanamines/butanamines_1983_BP.pdf Glennon RA, Young R, Jacyno JM, Slusher M, Rosecrans JA DOM-stimulus generalization to LSD and other hallucinogenic indolealkylamines Eur. J. Pharmacol., 1983, 86(3-4), 453-459 Medline (PMID=6572591) Young R, Rosecrans JA, Glennon RA Behavioral effects of 5-methoxy-N,N-dimethyltryptamine and dose-dependent antagonism by BC-105 Psychopharm. (Berl)., 1983, 80(2), 156-160 Medline (PMID=6410445) Kline TB, Benington F, Morin RD, Beaton JM, Glennon RA, Domelsmith LN, Houk KN, Rozeboom MD Structure-activity relationships for hallucinogenic N,N-dialkyltryptamines: photoelectron spectra and serotonin receptor affinities of methylthio and methylenedioxy derivatives J. Med. Chem., 1982, 25(11), 1381-1383 Medline (PMID=6815326) Glennon RA, Young R, Benington F, Morin RD Behavioral and serotonin receptor properties of 4-substituted derivatives of the hallucinogen 1-(2,5-dimethoxyphenyl)-2-aminopropane J. Med. Chem., 1982, 25(10), 1163-1168 Medline (PMID=7143352) https://www.rhodium.ws/pdf/glennon.4-pos-sar.dof-doi-don.pdf Glennon RA, Young R Comparison of behavioral properties of di- and tri-methoxyphenylisopropylamines Pharmacol. Biochem. Behav., 1982, 17(4), 603-607 Medline (PMID=6965276) Post 512438 (7is: "All the missing PBB articles part 1", General Discourse) Glennon RA, Gessner PK, Godse DD, Kline BJ Bufotenine esters J. Med. Chem., 1979, 22(11), 1414-1416 Medline (PMID=533890) Grella B, Dukat M, Young R, Teitler M, Herrick-Davis K, Gauthier CB, Glennon RA Investigation of hallucinogenic and related beta-carbolines Drug Alcohol Depend., 1998, 50(2), 99-107 Medline (PMID=9649961) Post 494854 (Nicodem: "Papers on beta-carbolines", General Discourse) Glennon RA Classical hallucinogens: an introductory overview NIDA Res Monogr., 1994, 146, 4-32 Medline (PMID=8742792) Glennon RA, Teitler M, Sanders-Bush E Hallucinogens and serotonergic mechanisms NIDA Res Monogr., 1992, 119, 131-135 Medline (PMID=1435968) Glennon RA Phenylalkylamine stimulants, hallucinogens, and designer drugs NIDA Res Monogr., 1991, 105, 154-160 Medline (PMID=1678860) Darmani NA, Martin BR, Pandey U, Glennon RA Pharmacological characterization of ear-scratch response in mice as a behavioral model for selective 5-HT2-receptor agonists and evidence for 5-HT1B- and 5-HT2-receptor interactions Pharmacol. Biochem. Behav., 1990, 37(1), 95-99 Medline (PMID=2263671) Post 512438 (7is: "All the missing PBB articles part 1", General Discourse) Glennon RA Stimulus properties of hallucinogenic phenalkylamines and related designer drugs: formulation of structure-activity relationships NIDA Res Monogr., 1989, 94, 43-67 Medline (PMID=2575229) Glennon RA, Titeler M, Lyon RA A preliminary investigation of the psychoactive agent 4-bromo-2,5-dimethoxyphenethylamine: a potential drug of abuse Pharmacol. Biochem. Behav., 1988, 30(3), 597-601 Medline (PMID=3211969) https://www.rhodium.ws/pdf/glennon.2c-b.pdf Glennon RA, Titeler M, Lyon RA, Slusher RM N,N-di-n-propylserotonin: binding at serotonin binding sites and a comparison with 8-hydroxy-2-(di-n-propylamino)tetralin J. Med. Chem., 1988, 31(4), 867-870 Medline (PMID=2965244) Titeler M, Herrick K, Lyon RA, McKenney JD, Glennon RA [3H]DOB: a specific agonist radioligand for 5-HT2 serotonin receptors Eur. J. Pharmacol., 1985, 117(1), 145-146 Medline (PMID=4085543) Glennon RA, Jacyno JM, Young R A comparison of the behavioral properties of (±)-, (-)-, and (+)-5-methoxy-alpha-methyltryptamine Biol. Psychiatry., 1983, 18(4), 493-498 Medline (PMID=6860723) Young R, Rosecrans JA, Glennon RA Comparative discriminative stimulus effects of 5-methoxy-N,N-dimethyltryptamine and LSD Life Sci., 1982, 30(24), 2057-2062 Medline (PMID=7109835) Post 508287 (not existing) Glennon RA, Young R, Rosecrans JA A comparison of the behavioral effects of DOM homologs Pharmacol. Biochem. Behav., 1982, 16(4), 557-559 Medline (PMID=7071089) Post 512438 (7is: "All the missing PBB articles part 1", General Discourse) Glennon RA, Young R, Rosecrans JA Discriminative stimulus properties of DOM and several molecular modifications Pharmacol. Biochem. Behav., 1982, 16(4), 553-536 Medline (PMID=7071088) Post 512438 (7is: "All the missing PBB articles part 1", General Discourse) Glennon RA, Young R, Benington F, Morin RD Hallucinogens as discriminative stimuli: a comparison of 4-OMe DMT and 5-OMe DMT with their methythio counterparts Life Sci., 1982, 30(5), 465-467 Medline (PMID=6801410) Post 508287 (not existing) Glennon RA, Rosecrans JA Indolealkylamine and phenalkylamine hallucinogens: a brief overview Neurosci. Biobehav. Rev., 1982, 6(4), 489-497 Medline (PMID=6757811) Glennon RA, Rosecrans JA, Young R Behavioral properties of psychoactive phenylisopropylamines in rats Eur. J. Pharmacol., 1981, 76(4), 353-360 Medline (PMID=7327208) Domelsmith LN, Eaton TA, Houk KN, Anderson GM 3rd, Glennon RA, Shulgin AT, Castagnoli N Jr, Kollman PA Photoelectron spectra of psychotropic drugs. 6. Relationships between the physical properties and pharmacological actions of amphetamine analogues J. Med. Chem., 1981, 24(12), 1414-1421 Medline (PMID=7310818) https://www.rhodium.ws/pdf/drugs.photoelectron.spectra-6.pdf Glennon RA, Doot DL, Young R DOM and related 2,5-dimethoxy-4-alkylphenylisopropylamines: behavioral and serotonin receptor properties Pharmacol. Biochem. Behav., 1981, 14(3), 287-292 Medline (PMID=7232455) Post 512466 (7is: "All the missing PBB articles part 2", General Discourse) Glennon RA, Rosecrans JA Speculations on the mechanism of action of hallucinogenic indolealkylamines Neurosci. Biobehav. Rev., 1981, 5(2), 197-207 Medline (PMID=7022271) Glennon RA, Liebowitz SM, Leming-Doot D, Rosecrans JA Demethyl analogues of psychoactive methoxyphenalkylamines: synthesis and serotonin receptor affinities J. Med. Chem., 1980, 23(9), 990-994 Medline (PMID=7411554) Glennon RA, Liebowitz SM, Anderson GM 3rd Serotonin receptor affinities of psychoactive phenalkylamine analogues J. Med. Chem., 1980, 23(3), 294-299 Medline (PMID=7365744) https://www.rhodium.ws/pdf/glennon.pea.receptor.affinities.pdf Minnema D, Krynock G, Young R, Glennon R, Rosecrans J LSD as a discriminative stimulus: role of dorsal raphe nucleus Subst Alcohol Actions Misuse., 1980, 1(1), 29-34 Medline (PMID=7323940) Young R, Glennon RA, Rosecrans JA Discriminative stimulus properties of the hallucinogenic agent DOM Commun. Psychopharmacol., 1980, 4(6), 501-506 Medline (PMID=7297054) Glennon RA, Young R, Rosecrans JA, Kallman MJ Hallucinogenic agents as discriminative stimuli: a correlation with serotonin receptor affinities Psychopharm. (Berl)., 1980, 68(2), 155-158 Medline (PMID=6776558) Glennon RA, Kier LB, Shulgin AT Molecular connectivity analysis of hallucinogenic mescaline analogs J. Pharm. Sci., 1979, 68(7), 906-907 Medline (PMID=458614) https://www.rhodium.ws/pdf/shulgin/shulgin.molecular.connectivity.pdf Glennon RA, Gessner PK Serotonin receptor binding affinities of tryptamine analogues J. Med. Chem., 1979, 22(4), 428-432 Medline (PMID=430481) Glennon RA, Rosecrans JA, Young R, Gaines J Hallucinogens as a discriminative stimuli: generalization of DOM to a 5-methoxy-N, N-dimethyltryptamine stimulus Life Sci., 1979, 24(11), 993-997 Medline (PMID=286864) Post 508287 (not existing) Glennon RA, Liebowitz SM, Mack EC Serotonin receptor binding affinities of several hallucinogenic phenylalkylamine and N,N-dimethyltryptamine analogues J. Med. Chem., 1978, 21(8), 822-825 Medline (PMID=278843) (Uploaded file not existing) Kier LB, Glennon RA Psychotomimetic phenalkylamines as serotonin agonists: an SAR analysis Life Sci., 1978, 22(18), 1589-1593 Medline (PMID=672414) Post 508287 (not existing) Kier LB, Glennon RA Progress with several models for the study of the SAR of hallucinogenic agents NIDA Res. Monogr., 1978, (22), 159-185 Medline (PMID=101879) Glennon RA, Gessner PK The electronic and serotonin receptor binding affinity properties of N,N-dimethyltryptamine analogs Res. Commun. Chem. Pathol. Pharmacol., 1977, 18(3), 453-465 Medline (PMID=270770) Glennon RA A quantum chemical investigation of the pi-electronic structure of the hallucinogenic N,N-dimethyltryptamines Res. Commun. Chem. Pathol. Pharmacol., 1974, 9(1), 185-188 Medline (PMID=4531086) Glennon, R. A.; Kier, L. B LSD Analogs as serotonin antagonists: A molecular connectivity SAR analysis Eur. J. Med. Chem., 1978, 13, 219 No PubMed entry or DOI found Minnema, D.; Krynock, G.; Young, R.; Glennon, R. A.; Rosecrans, J. A Role of dorsal raphe neurons to the ability of LSD to act as a discriminative stimulus J. Alcohol Drug Abuse, 1980, 1, 29 No PubMed entry or DOI found Westkaemper, R.B.; Dukat, M.; Glennon, R.A Molecular modeling of drug-receptor interactions using a 5-HT2 receptor model Med. Chem. Res., 1991, 1, 401-408 No PubMed entry or DOI found Westkaemper, R.B. and Glennon, R.A Molecular graphics models of members of the 5-HT2 subfamily: 5-HT2A, 5-HT2B, and 5-HT2C receptors Med. Chem. Res., 1993, 3, 317-334 No PubMed entry or DOI found Carroll, F.I.; Glennon, R.A.; Johnson, M.R.; Teitler, M.; Zimmerman, D. M Hallucinogenic Agents: Drugs of abuse as neurochemical tools NIDA Res. Mono., 1994, 140, 94-98 No PubMed entry or DOI found Dukat, M.; Herrick-Davis, K.; Teitler, M.; Glennon, R.A Piperidine derivatives of serotonin as selective 5-HT1A serotonin receptor agonists Med. Chem. Res., 1994, 4, 254-258 No PubMed entry or DOI found Ismaiel, A.M. Dukat, M., Nelson, D.L. Lucaites, V.L.; Glennon, R.A Binding of N2-substituted pyrio[4,3-b]indole analogs of spiperone at human 5-HT2A, 5-HT2B, and 5-HT2C serotonin receptors Med. Chem. Res., 1996, 6, 197-211 No PubMed entry or DOI found Malmusi, L.; Dukat, M.; Young, R.; Teitler, M.; Darmani, N.; Ahmad, B.; Smith, C.; Glennon, R. A 1,2,3,4- Tetrahydroisoquinolines and related analogs of the phenylalkylamine stimulants and hallucinogens Med. Chem. Res. 1996, 6, 400-411 No PubMed entry or DOI found Glennon, R. A.; Dukat, M Novel serotonergic agents: 5-HT2 – Update 1997 Investigational Drugs Research Alerts, 1997, 2, 107-113 No PubMed entry or DOI found Westkaemper, R. B.; Hyde, E. G.; Choudhary, M. S.; Khan, N.; Gelbar, E.; Glennon, R. A.; Roth, B. L Engineering a region of bulk tolerance in the 5-HT2A receptor Eur. J. Med. Chem., 1999, 34, 441-447 No PubMed entry or DOI found Khorana, N.; Bondarev, M.; Dukat, M.; Herrick-Davis, K.; Egan, C.; DuPre, A.; Smith, C.; Teitler, M.; Glennon, R. A Binding of spiperone analogs at 5-HT2A serotonin receptors Med. Chem. Res., 1999, 9, 657-667 No PubMed entry or DOI found Hong, S.; Dukat, M.; Teitler, M.; Egan, C.; DuPre, A.; Herrick-Davis, K.; Glennon, R. A 5,8-Dimethoxyharmalan: Actions at 5-HT2A serotonin receptors Med. Chem. Res., 1999, 9, 374-388 No PubMed entry or DOI found Glennon RA Arylalkylamine drugs of abuse: an overview of drug discrimination studies Pharmacol. Biochem. Behav., 1999, 64(2), 251-256 Medline (PMID=10515299) https://www.rhodium.ws/pdf/glennon.arylalkylamine.drugs.of.abuse.pdf Darmani NA, Martin BR, Glennon RA Behavioral evidence for differential adaptation of the serotonergic system after acute and chronic treatment with (+/-)-1-(2,5-dimethoxy-4-iodophenyl)-2-aminopropane (DOI) or ketanserin J. Pharmacol. Exp. Ther., 1992, 262(2), 692-698 Medline (PMID=1501117) Glennon RA Discriminative stimulus properties of hallucinogens and related designer drugs NIDA Res. Monogr., 1991, (116), 25-44 Medline (PMID=1369672) Higgs RA, Glennon RA Stimulus properties of ring-methyl amphetamine analogs Pharmacol. Biochem. Behav., 1990, 37(4), 835-837 Medline (PMID=2093186) Post 512466 (7is: "All the missing PBB articles part 2", General Discourse) Nichols DE, Glennon RA Medicinal chemistry and structure-activity relationships of hallucinogens. In: Jacobs, B.L., ed. Hallucinogens: Neurochemical, Behavioral, and Clinical Perspectives. New York: Raven Press, 1984. pp. 95-142 No PubMed entry or DOI found Ligands of other 5-HT receptor subtypes Pullagurla MR, Westkaemper RB, Glennon RA Possible differences in modes of agonist and antagonist binding at human 5-HT6 receptors Bioorg. Med. Chem. Lett., 2004, 14(17), 4569-4573 Medline (PMID=15357994) Prisinzano T, Dukat M, Law H, Slassi A, MacLean N, DeLannoy I, Glennon RA 2-(Anilino)imidazolines and 2-(benzyl)imidazoline derivatives as h5-HT1D serotonin receptor ligands Bioorg. Med. Chem. Lett., 2004, 14(18), 4697-4699 Medline (PMID=15324890) Dukat M, Smith C, Herrick-Davis K, Teitler M, Glennon RA Binding of tryptamine analogs at h5-HT1E receptors: a structure-affinity investigation Bioorg. Med. Chem., 2004, 12(10), 2545-2552 Medline (PMID=15110837) Chang-Fong J, Rangisetty JB, Dukat M, Setola V, Raffay T, Roth B, Glennon RA 1,2,3,4-tetrahydrocarbazoles as 5-HT6 serotonin receptor ligands Bioorg. Med. Chem. Lett., 2004, 14(8), 1961-1964 Medline (PMID=15050637) Glennon RA, Daoud MK, Dukat M, Teitler M, Herrick-Davis K, Purohit A, Syed H Arylguanidine and arylbiguanide binding at 5-HT3 serotonin receptors: a QSAR study Bioorg. Med. Chem., 2003, 11(20), 4449-4454 Medline (PMID=13129581) Pullagurla MR, Dukat M, Setola V, Roth B, Glennon RA N1-benzenesulfonylgramine and N1-benzenesulfonylskatole: novel 5-HT6 receptor ligand templates Bioorg. Med. Chem. Lett., 2003, 13(19), 3355-3359 Medline (PMID=12951125) Khorana N, Smith C, Herrick-Davis K, Purohit A, Teitler M, Grella B, Dukat M, Glennon RA Binding of tetrahydrocarboline derivatives at human 5-HT5A receptors J. Med. Chem., 2003, 46(18):3930-3937 Medline (PMID=12930153) Glennon RA Higher-end serotonin receptors: 5-HT5, 5-HT6, and 5-HT7 J. Med. Chem., 2003, 46(14), 2795-2812 Medline (PMID=12825922) Rahman AA, Daoud MK, Dukat M, Herrick-Davis K, Purohit A, Teitler M, do Amaral AT, Malvezzi A, Glennon RA Conformationally-restricted analogues and partition coefficients of the 5-HT3 serotonin receptor ligands meta-chlorophenylbiguanide (mCPBG) and meta-chlorophenylguanidine (mCPG) Bioorg. Med. Chem. Lett., 2003, 13(6):1119-1123 Medline (PMID=12643925) Khorana N, Purohit A, Herrick-Davis K, Teitler M, Glennon RA gamma-Carbolines: binding at 5-HT5A serotonin receptors Bioorg. Med. Chem., 2003, 11(5), 717-722 Medline (PMID=12538001) Runyon SP, Peddi S, Savage JE, Roth BL, Glennon RA, Westkaemper RB Geometry-affinity relationships of the selective serotonin receptor ligand 9-(aminomethyl)-9,10-dihydroanthracene J. Med. Chem., 2002, 45(8), 1656-1664 Medline (PMID=11931619) Dukat M, Choi YN, Teitler M, Du Pre A, Herrick-Davis K, Smith C, Glennon RA The binding of arylguanidines at 5-HT3 serotonin receptors: a structure-affinity investigation Bioorg. Med. Chem. Lett., 2001, 11(12), 1599-1603 Medline (PMID=11412989) Prisinzano T, Law H, Dukat M, Slassi A, MaClean N, Demchyshyn L, Glennon RA Imidazoline-modified benzylimidazolines as h5-HT1D/1B serotonergic ligands Bioorg. Med. Chem., 2001, 9(3):613-619 Medline (PMID=11310595) Runyon SP, Savage JE, Taroua M, Roth BL, Glennon RA, Westkaemper RB Influence of chain length and N-alkylation on the selective serotonin receptor ligand 9-(aminomethyl)-9,10-dihydroanthracene Bioorg. Med. Chem. Lett., 2001, 11(5), 655-658 Medline (PMID=11266163) Westkaemper RB, Runyon SP, Savage JE, Roth BL, Glennon RA Exploring the relationship between binding modes of 9-(aminomethyl)-9,10-dihydroanthracene and cyproheptadine analogues at the 5-HT2A serotonin receptor Bioorg. Med. Chem. Lett., 2001, 11(4), 563-566 Medline (PMID=11229772) Tsai Y, Dukat M, Slassi A, MacLean N, Demchyshyn L, Savage JE, Roth BL, Hufesein S, Lee M, Glennon RA N1-(Benzenesulfonyl)tryptamines as novel 5-HT6 antagonistst Bioorg. Med. Chem. Lett., 2000, 10(20), 2295-2299 Medline (PMID=11055342) Dukat M, Young R, Darmani NN, Ahmed B, Glennon RA The 5-HT3 agent N-(3-chlorophenyl)guanidine (MD-354) serves as a discriminative stimulus in rats and displays partial agonist character in a shrew emesis assay Psychopharm. (Berl)., 2000, 150(2), 200-207 Medline (PMID=10907673) Glennon RA, Lee M, Rangisetty JB, Dukat M, Roth BL, Savage JE, McBride A, Rauser L, Hufeisen S, Lee DK 2-Substituted tryptamines: agents with selectivity for 5-HT6 serotonin receptors J. Med. Chem., 2000, 43(5), 1011-1018 Medline (PMID=10715164) http://pharmacist8.tripod.com/2-subst-trypt.pdf Law H, Dukat M, Teitler M, Lee DK, Mazzocco L, Kamboj R, Rampersad V, Prisinzano T, Glennon RA Benzylimidazolines as h5-HT1B/1D serotonin receptor ligands: a structure-affinity investigation J. Med. Chem., 1998, 41(13), 2243-2251 Medline (PMID=9632357) Ismaiel AM, Dukat M, Law H, Kamboj R, Fan E, Lee DK, Mazzocco L, Buekschkens D, Teitler M, Pierson ME, Glennon RA 2-(1-Naphthyloxy)ethylamines with enhanced affinity for human 5-HT1D beta (h5-HT1B) serotonin receptors J. Med. Chem., 1997, 40(26), 4415-4419 Medline (PMID=9435911) Dukat M, Abdel-Rahman AA, Ismaiel AM, Ingher S, Teitler M, Gyermek L, Glennon RA Structure-activity relationships for the binding of arylpiperazines and arylbiguanides at 5-HT3 serotonin receptors J. Med. Chem., 1996, 39(20), 4017-4026 Medline (PMID=8831767) https://www.rhodium.ws/pdf/glennon.arylpiperazines.5ht3.pdf Glennon RA, Hong SS, Bondarev M, Law H, Dukat M, Rakhi S, Power P, Fan E, Kinneau D, Kamboj R, Teitler M, Herrick-Davis K, Smith C Binding of O-alkyl derivatives of serotonin at human 5-HT1D beta receptors J. Med. Chem., 1996, 39(1), 314-322 Medline (PMID=8568822) Glennon RA, Hong SS, Dukat M, Teitler M, Davis K 5-(Nonyloxy)tryptamine: a novel high-affinity 5-HT1D beta serotonin receptor agonist J. Med. Chem., 1994, 37(18), 2828-2830 Medline (PMID=8071931) Glennon RA, Young R, Dukat M 5-HT3 agonist 2-methylserotonin as a training drug in discrimination studies Pharmacol. Biochem. Behav., 1992, 41(2), 361-364 Medline (PMID=1574526) Post 512466 (7is: "All the missing PBB articles part 2", General Discourse) Westkaemper RB, Glennon RA Approaches to molecular modeling studies and specific application to serotonin ligands and receptors Pharmacol. Biochem. Behav., 1991, 40(4), 1019-1031 Medline (PMID=1816556) Post 512466 (7is: "All the missing PBB articles part 2", General Discourse) Glennon RA, Dukat M Serotonin receptors and their ligands: a lack of selective agents Pharmacol. Biochem. Behav., 1991, 40(4), 1009-1017 Medline (PMID=1816555) Post 512466 (7is: "All the missing PBB articles part 2", General Discourse) Raghupathi RK, Rydelek-Fitzgerald L, Teitler M, Glennon RA Analogues of the 5-HT1A serotonin antagonist 1-(2-methoxyphenyl)-4-[4-(2-phthalimido)butyl]piperazine with reduced alpha 1-adrenergic affinity J. Med. Chem., 1991, 34(8), 2633-2638 Medline (PMID=1652026) Glennon RA Serotonin receptors and site-selective agents J. Physiol. Pharmacol., 1991, 42(1), 49-60 Medline (PMID=1932772) Glennon RA, Darmani NA, Martin BR Multiple populations of serotonin receptors may modulate the behavioral effects of serotonergic agents Life Sci., 1991, 48(26), 2493-2498 Medline (PMID=2046474) Post 508288 (7is: "All the missing Life Sciences articles part 2", General Discourse) Rydelek-Fitzgerald L, Teitler M, Fletcher PW, Ismaiel AM, Glennon RA NAN-190: agonist and antagonist interactions with brain 5-HT1A receptors Brain Res., 1990, 532(1-2), 191-196 Medline (PMID=2282513) Ismaiel AM, Titeler M, Miller KJ, Smith TS, Glennon RA 5-HT1 and 5-HT2 binding profiles of the serotonergic agents alpha-methylserotonin and 2-methylserotonin J. Med. Chem., 1990, 33(2), 755-758 Medline (PMID=2299641) Glennon RA Serotonin receptors: clinical implications Neurosci. Biobehav. Rev., 1990, 14(1), 35-47 Medline (PMID=2183098) Glennon RA, Ismaiel AE, McCarthy BG, Peroutka SJ Binding of arylpiperazines to 5-HT3 serotonin receptors: results of a structure-affinity study Eur. J. Pharmacol., 1989, 168(3), 387-392 Medline (PMID=2583244) Glennon RA, Naiman NA, Pierson ME, Smith JD, Ismaiel AM, Titeler M, Lyon RA N-(phthalimidoalkyl) derivatives of serotonergic agents: a common interaction at 5-HT1A serotonin binding sites? J. Med. Chem., 1989, 32(8), 1921-1926 Medline (PMID=2754715) Pierson ME, Lyon RA, Titeler M, Schulman SB, Kowalski P, Glennon RA Design and synthesis of propranolol analogues as serotonergic agents J. Med. Chem., 1989, 32(4), 859-863 Medline (PMID=2539480) Naiman N, Lyon RA, Bullock AE, Rydelek LT, Titeler M, Glennon RA 2-(Alkylamino)tetralin derivatives: interaction with 5-HT1A serotonin binding sites J. Med. Chem., 1989, 32(1), 253-256 Medline (PMID=2521252) Glennon RA, Naiman NA, Lyon RA, Titeler M Arylpiperazine derivatives as high-affinity 5-HT1A serotonin ligands J. Med. Chem., 1988, 31(10), 1968-1971 Medline (PMID=3172131) Glennon RA, Naiman NA, Pierson ME, Titeler M, Lyon RA, Weisberg E NAN-190: an arylpiperazine analog that antagonizes the stimulus effects of the 5-HT1A agonist 8-hydroxy-2-(di-n-propylamino)tetralin (8-OH-DPAT) Eur. J. Pharmacol., 1988, 154(3), 339-341 Medline (PMID=2976673) Glennon RA Site-selective serotonin agonists as discriminative stimuli Psychopharmacol. Ser., 1988, 4, 15-31 Medline (PMID=3293039) Glennon RA Central serotonin receptors as targets for drug research J. Med. Chem., 1987, 30(1), 1-12 Medline (PMID=3543362) Lyon RA, Titeler M, McKenney JD, Magee PS, Glennon RA Synthesis and evaluation of phenyl- and benzoylpiperazines as potential serotonergic agents J. Med. Chem., 1986, 29(5), 630-634 Medline (PMID=3701781) McKenney JD, Glennon RA TFMPP may produce its stimulus effects via a 5-HT1B mechanism Pharmacol. Biochem. Behav., 1986, 24(1), 43-47 Medline (PMID=3945665) Arvidsson LE, Hacksell U, Glennon RA Recent advances in central 5-hydroxytryptamine receptor agonists and antagonists Prog. Drug. Res., 1986, 30, 365-471 Medline (PMID=3544048) Glennon RA, McKenney JD, Young R Discriminative stimulus properties of the serotonin agonist 1-(3-trifluoromethylphenyl)piperazine (TFMPP) Life Sci., 1984, 35(14), 1475-1480 Medline (PMID=6482668) Post 508287 (not existing) Glennon RA, Young R, Rosecrans JA Antagonism of the effects of the hallucinogen DOM and the purported 5-HT agonist quipazine by 5-HT2 antagonists Eur. J. Pharmacol., 1983, 91(2-3), 189-96 Medline (PMID=6617740) Glennon RA, Jacyno JM, Salley JJ Jr 2,3-dihydro and carbocyclic analogues of tryptamines: interaction with serotonin receptors J. Med. Chem., 1982, 25(1), 68-70 Medline (PMID=7086824) Glennon RA Serotonin receptor interactions of harmaline and several related beta-carbolines Life Sci., 1981, 29(8), 861-865 Medline (PMID=7300579) Post 508287 (not existing) Glennon RA The effect of chirality on serotonin receptor affinity Life Sci., 1979, 24(16), 1487-1492 Medline (PMID=470548) Post 508287 (not existing) Glennon RA, Martin B, Johnson KM, End D 7,N,N-Trimethyltryptamine: a selective inhibitor of synaptosomal serotonin uptake Res. Commun. Chem. Pathol. Pharmacol., 1978, 19(1), 161-164 Medline (PMID=625585) Glennon, R. A.; Naiman, N. A.; Pierson, M. E.; Titeler, M.; Lyon, R. A.; Herndon, J. L.; Misenheimer, B Stimulus properties of arylpiperazines: NAN-190, a potential 5-HT1A serotonin antagonist Drug. Dev. Res., 1989, 16, 335-343 No PubMed entry or DOI found Ismaiel, A. M.; Titeler, M.; Glennon, R. A g-Carboline derivatives as potential serotonergic agents Mansoura J. Pharm. (Egypt) 1989, 6, 1-13 No PubMed entry or DOI found Glennon, R. A., Raghupathi, R. K Serotonin receptor ligands Current CNS Patents 1990, 1, 323-343 No PubMed entry or DOI found Glennon, R.A Serotonin receptors and site-selective agents J. Physiol. Pharmacol. (Poland) 1991, 1, 42-60 No PubMed entry or DOI found Glennon, R. A., Ismaiel, A. M., Chaurasia, C., Titeler, M 5-HT1D serotonin receptors: Results of a structure- affinity investigation Drug Dev. Res. 1991, 22, 25-36 No PubMed entry or DOI found Glennon, R.A., El-Ashmawy, M., Ismaiel, A.M., Fischer, J.B Binding of N-substituted 2-phenylaminoethanes to s and serotonin 5-HT1A receptors Med. Chem. Res., 1991, 1, 109-114 No PubMed entry or DOI found Glennon, R.A., Bartyzel, P., Teitler, M Binding of benz[e]-and benz[g]-fused tryptamine derivatives at serotonin receptors: Evidence for a region of bulk tolerance Med. Chem. Res., 1991, 1, 201-206 No PubMed entry or DOI found Glennon, R. A.; Darmani, N.; Martin, W Modulation of the behavioral effects of serotonergic agents by multiple 5-HT receptors Life Sci., 1991, 48, 2493-2498 No PubMed entry or DOI found Dukat, M.; Miller, K.; Teitler, M.; Glennon, R.A Binding of amine-substituted and quaternary amine analogs of serotonin at 5-HT3 serotonin receptors Med. Chem. Res., 1991, 1, 271-276 No PubMed entry or DOI found Bakthavachalam, V.; Fell, B.; Teitler, M.; Glennon, R.A.; Neumeyer, J.L Fluorescent probes for serotonin 5-HT1A receptors: synthesis, receptor affinity and selectivity Med. Chem. Res., 1991, 1, 265-270 No PubMed entry or DOI found Glennon, R.A Preface for special serotonin issue Pharmacol. Biochem. Behav., 1991, 40, 1007 No PubMed entry or DOI found El-Bermawy, M.; Raghupathi, R.; Ingher, S. P.; Teitler, M.; Maayani, S.; Glennon, R. A 4-[4-(1-Noradamantane carboxamido)butyl]-1-(2-methoxyphenyl) piperazine: A high affinity 5-HT1A-selective agent Med. Chem. Res., 1992, 2, 88-95 No PubMed entry or DOI found El-Bermawy, M.; Lotter, H.; Glennon, R.A Comparative molecular field analysis of the binding of arylpiperazines at 5-HT1A serotonin receptors Med. Chem. Res., 1992, 2, 290-297 No PubMed entry or DOI found Glennon, R.A Concepts for design of 5-HT1A serotonin agonists and antagonists Drug Dev. Res., 1992, 26, 251-274 No PubMed entry or DOI found Westkaemper, R.B.; Yousif, M.; Teitler, M.; Glennon, R.A Binding of aporphines at 5-HT1A serotonin receptors: A computational investigation of potential binding modes Med. Chem. Res., 1992, 2, 482-490 No PubMed entry or DOI found Glennon, R.A.; Dukat, M 5-HT receptor ligands: Update 1992 Current Drugs, 1992, 1, 1-45 No PubMed entry or DOI found Glennon, R.A., Westkaemper, R.B 5-HT1D Receptors: A serotonin receptor population for the 1990s Drug News Perspect., 1993, 6, 390-405 No PubMed entry or DOI found Hong, S.-S.; Dukat, M.; Teitler, M.; Herrick-Davis, K.; McCallum, K.; Kamboj, R.; Glennon, R.A Binding of 5-arylalkyloxytryptamines at human 5-HT1Dß serotonin receptors Med. Chem. Res., 1995, 5, 690-699 No PubMed entry or DOI found Iwamura, T.; Casey, C. T.; Young, R.; Dukat, M.; Teitler, M.; Fadden, J. S. P.; Glennon, R. A 4-(6-Fluorobenzisoxazol-3-yl)piperidine, a risperidone metabolite with serotonergic activity of potential clinical significance Med. Chem. Res., 1996, 6, 593-601 No PubMed entry or DOI found Glennon, R. A.; Dukat, M 5-HT1 receptor ligands: Update 1997 Investigational Drugs Research Alerts, 1997, 2, 351-372 No PubMed entry or DOI found Teitler, M.; Schieck, C.; Howard, P.; Sullivan, J. E.; Iwamura, T.; Glennon, R. A 5-HT5A serotonin receptors: A preliminary structure-affinity investigation Med. Chem. Res., 1997, 7, 207-218 No PubMed entry or DOI found Bondarev, M.; Iwamura, T.; Hynd, D.; Mazzocco, L.; Lee, D. K. H.; Dukat, M.; Glennon, R. A Aryloxyethylamines as h5-HT1D serotonin receptor ligands Med. Chem. Res., 1998, 8, 333-342 No PubMed entry or DOI found Glennon, R. A.; Bondarev, M.; Roth, B 5-HT6 serotonin receptor binding of indolealkylamines: A preliminary structure-affinity investigation Med. Chem. Res., 1999, 9, 108-117 No PubMed entry or DOI found Lee, M.; Rangisetty, J. B.; Dukat, M.; Slassi, A.; McClean, N.; Lee, D. K. H.; Glennon, R. A 5-HT6 serotonin receptor binding affinities of N1-benzenesulfonyl and related tryptamines Med. Chem. Res., 2000, 10, 230-242 No PubMed entry or DOI found Prisinzano, T.; Law, H.; Slassi, A.; Maclean, N.; Demchyshyn, L.; Glennon, R. A QSAR studies on 2-(benzyl)imidazoline analogs as 5-HT1B/1D serotonin receptor ligands Med. Chem. Res., 2001, 10, 309-317 No PubMed entry or DOI found Wood PL, Pilapil C, LaFaille F, Nair NP, Glennon RA Unique [3H]tryptamine binding sites in rat brain: distribution and pharmacology Arch. Int. Pharmacodyn. Ther., 1984, 268(2), 194-201 Medline (PMID=6732364) Jeffery LH, Glennon RA Serotonin Receptors, Agents, and Actions In Drug Design for Neuroscience. ed. Alan P. Kozikowski., Raven Press. Ltd., New York 1993, 167-212 No PubMed entry or DOI found Stimulants: synthesis and pharmacology (MDMA, MDA, PMMA, (meth)ampehtamine, cathinone, ephedrine, etc.) Pullagurla M, Bondareva T, Young R, Glennon RA Modulation of the stimulus effects of (+)amphetamine by the 5-HT(6) antagonist MS-245 Pharmacol. Biochem. Behav., 2004, 78(2), 263-268 Medline (PMID=15219766) Khorana N, Pullagurla MR, Young R, Glennon RA Comparison of the discriminative stimulus effects of 3,4-methylenedioxymethamphetamine (MDMA) and cocaine: asymmetric generalization Drug Alcohol. Depend., 2004, 74(3), 281-287 Medline (PMID=15194206) Rothman RB, Vu N, Partilla JS, Roth BL, Hufeisen SJ, Compton-Toth BA, Birkes J, Young R, Glennon RA In vitro characterization of ephedrine-related stereoisomers at biogenic amine transporters and the receptorome reveals selective actions as norepinephrine transporter substrates J. Pharmacol. Exp. Ther., 2003, 307(1), 138-145 Medline (PMID=12954796) DOI:10.1124/jpet.103.053975 Post 509509 (Red_Crown: "Pharmacology of Ephedrine-related stereoisomers", Stimulants) Setola V, Hufeisen SJ, Grande-Allen KJ, Vesely I, Glennon RA, Blough B, Rothman RB, Roth BL 3,4-methylenedioxymethamphetamine (MDMA, "Ecstasy") induces fenfluramine-like proliferative actions on human cardiac valvular interstitial cells in vitro Mol. Pharmacol., 2003, 63(6), 1223-1229 Medline (PMID=12761331) Bondareva TS, Young R, Glennon RA Central stimulants as discriminative stimuli. Asymmetric generalization between (-)ephedrine and S(+)methamphetamine Pharmacol. Biochem. Behav., 2002, 74(1),157-162 Medline (PMID=12376163) Post 512466 (7is: "All the missing PBB articles part 2", General Discourse) Glennon RA, Young R Effect of 1-(3,4-methylenedioxyphenyl)-2-aminopropane and its optical isomers in PMMA-trained rats Pharmacol. Biochem. Behav., 2002, 72(1-2), 307-311 Medline (PMID=11900801) Post 512466 (7is: "All the missing PBB articles part 2", General Discourse) Dukat M, Young R, Glennon RA Effect of PMA optical isomers and 4-MTA in PMMA-trained rats Pharmacol. Biochem. Behav., 2002, 72(1-2), 299-305 Medline (PMID=11900800) Post 512466 (7is: "All the missing PBB articles part 2", General Discourse) Young R, Glennon RA The stimulus effect of 5,6,7,8-tetrahydro-1,3-dioxolo[4,5-g]isoquinoline is similar to that of cocaine but different from that of amphetamine Pharmacol. Biochem. Behav., 2002, 71(1-2), 205-213 Medline (PMID=11812524) http://www.maps.org/w3pb/new/2002/2002_young_1325_1.pdf Hong SS, Young R, Glennon RA Discriminative stimulus properties of alpha-ethyltryptamine optical isomers Pharmacol. Biochem. Behav., 2001, 70(2-3), 311-316 Medline (PMID=11701202) https://www.rhodium.ws/pdf/alpha-ethyltryptamine.optical.isomers.pdf Rangisetty JB, Bondarev ML, Chang-Fong J, Young R, Glennon RA PMMA-stimulus generalization to the optical isomers of MBDB and 3,4-DMA Pharmacol. Biochem. Behav., 2001, 69(1-2), 261-267 Medline (PMID=11420094) Post 512466 (7is: "All the missing PBB articles part 2", General Discourse) Young R, Glennon RA Stimulus effects of phenylpropanolamine optical isomers in (+)amphetamine-trained rats Pharmacol. Biochem. Behav., 2000, 66(3), 489-494 Medline (PMID=10899360) Post 512466 (7is: "All the missing PBB articles part 2", General Discourse) Glennon RA, Young R MDMA stimulus generalization to the 5-HT1A serotonin agonist 8-hydroxy-2-(di-n-propylamino)tetralin Pharmacol. Biochem. Behav., 2000, 66(3), 483-438 Medline (PMID=10899359) Post 512466 (7is: "All the missing PBB articles part 2", General Discourse) Glennon RA, Young R (+)Amphetamine-stimulus generalization to an herbal ephedrine product Pharmacol. Biochem. Behav., 2000, 65(4), 655-658 Medline (PMID=10764918) Post 512562 (7is: "All the missing PBB articles part 3", General Discourse) Young R, Bondarev M, Glennon RA An examination of isomeric phenylpropanolamines in (-)ephedrine-trained rats Drug Alcohol Depend., 1999, 57(1), 1-6 Medline (PMID=10617308) Young R, Dukat M, Malmusi L, Glennon RA Stimulus properties of PMMA: effect of optical isomers and conformational restriction Pharmacol. Biochem. Behav., 1999, 64(2), 449-453 Medline (PMID=10515329) Post 512562 (7is: "All the missing PBB articles part 3", General Discourse) Young R, Glennon RA Discriminative stimulus effects of S(-)-methcathinone (CAT): a potent stimulant drug of abuse Psychopharm. (Berl)., 1998, 140(3), 250-256 Medline (PMID=9877004) Young R, Gabryszuk M, Glennon RA (-)Ephedrine and caffeine mutually potentiate one another's amphetamine-like stimulus effects Pharmacol. Biochem. Behav., 1998, 61(2), 169-173 Medline (PMID=9738532) Post 512562 (7is: "All the missing PBB articles part 3", General Discourse) Young R, Glennon RA Discriminative stimulus properties of (-)ephedrine Pharmacol. Biochem. Behav., 1998, 60(3), 771-775 Medline (PMID=9678664) Post 512562 (7is: "All the missing PBB articles part 3", General Discourse) Dal Cason TA, Young R, Glennon RA Cathinone: an investigation of several N-alkyl and methylenedioxy-substituted analogs Pharmacol. Biochem. Behav., 1997, 58(4), 1109-1116 Medline (PMID=9408221) https://www.rhodium.ws/pdf/cathinone-methylone.pdf Glennon RA, Young R, Dukat M, Cheng Y Initial characterization of PMMA as a discriminative stimulus Pharmacol. Biochem. Behav., 1997, 57(1-2), 151-158 Medline (PMID=9164566) Post 512562 (7is: "All the missing PBB articles part 3", General Discourse) Young R, Glennon RA Cocaine-stimulus generalization to MDA optical isomers: a reevaluation Pharmacol. Biochem. Behav., 1997, 57(1-2), 115-118 Medline (PMID=9164561) Post 512562 (7is: "All the missing PBB articles part 3", General Discourse) Young R, Darmani NA, Elder EL, Dumas D, Glennon RA Clobenzorex: evidence for amphetamine-like behavioral actions Pharmacol. Biochem. Behav., 1997, 56(2), 311-316 Medline (PMID=9050090) Post 512562 (7is: "All the missing PBB articles part 3", General Discourse) Young R, Glennon RA A three-lever operant procedure differentiates the stimulus effects of R(-)-MDA from S(+)-MDA J. Pharmacol. Exp. Ther., 1996, 276(2), 594-601 Medline (PMID=8632326) Glennon RA, Young R, Martin BR, Dal Cason TA Methcathione ("cat"): an enantiomeric potency comparison Pharmacol. Biochem. Behav., 1995, 50(4), 601-606 Medline (PMID=7617707) Post 512562 (7is: "All the missing PBB articles part 3", General Discourse) Glennon RA MDMA-like stimulus effects of alpha-ethyltryptamine and the alpha-ethyl homolog of DOM Pharmacol. Biochem. Behav., 1993, 46(2), 459-462 Medline (PMID=7903460) https://www.rhodium.ws/pdf/butanamines/butanamines_1993_PBB.pdf Young R, Glennon RA Cocaine-stimulus generalization to two new designer drugs: methcathinone and 4-methylaminorex Pharmacol. Biochem. Behav., 1993, 45(1), 229-231 Medline (PMID=8516363) Post 512562 (7is: "All the missing PBB articles part 3", General Discourse) Glennon RA, Higgs R, Young R, Issa H Further studies on N-methyl-1(3,4-methylenedioxyphenyl)-2-aminopropane as a discriminative stimulus: antagonism by 5-hydroxytryptamine3 antagonists Pharmacol. Biochem. Behav., 1992, 43(4), 1099-1106 Medline (PMID=1361990) Post 512562 (7is: "All the missing PBB articles part 3", General Discourse) Glennon RA, Higgs R Investigation of MDMA-related agents in rats trained to discriminate MDMA from saline Pharmacol. Biochem. Behav., 1992, 43(3), 759-763 Medline (PMID=1360162) Post 512562 (7is: "All the missing PBB articles part 3", General Discourse) Herndon JL, Pierson ME, Glennon RA Mechanistic investigation of the stimulus properties of 1-(3-trifluoromethylphenyl)piperazine Pharmacol. Biochem. Behav., 1992, 43(3), 739-748 Medline (PMID=1333084) Post 512563 (7is: "All the missing PBB articles part 4", General Discourse) Yousif MY, Fitzgerald RL, Narasimhachari N, Rosecrans JA, Blanke RV, Glennon RA Identification of metabolites of 3,4-methylenedioxymethamphetamine in rats Drug Alcohol Depend., 1990, 26(2), 127-135 Medline (PMID=1978707) Glennon RA, Misenheimer B Stimulus properties of a new designer drug: 4-methylaminorex ("U4Euh") Pharmacol. Biochem. Behav., 1990, 35(3), 517-521 Medline (PMID=1971111) Post 512563 (7is: "All the missing PBB articles part 4", General Discourse) Teitler M, Leonhardt S, Appel NM, De Souza EB, Glennon RA Receptor pharmacology of MDMA and related hallucinogens Ann N Y Acad Sci., 1990, 600, 626-38, discussion 638-639 Medline (PMID=1979215) Glennon RA, Misenheimer BR Stimulus effects of N-monoethyl-1-(3,4-methylenedioxyphenyl)-2-aminopropane (MDE) and N-hydroxy-1-(3,4-methylenedioxyphenyl)-2-aminopropane (N-OH MDA) in rats trained to discriminate MDMA from saline Pharmacol. Biochem. Behav., 1989, 33(4), 909-912 Medline (PMID=2575759) Post 512563 (7is: "All the missing PBB articles part 4", General Discourse) Fitzgerald RL, Blanke RV, Glennon RA, Yousif MY, Rosecrans JA, Poklis A Determination of 3,4-methylenedioxyamphetamine and 3,4-methylenedioxymethamphetamine enantiomers in whole blood J. Chromatogr., 1989, 490(1), 59-69 Medline (PMID=2760158) Fitzgerald RL, Blanke RV, Rosecrans JA, Glennon RA Stereochemistry of the metabolism of MDMA to MDA Life Sci., 1989, 45(4), 295-301 Medline (PMID=2569654) Post 508288 (7is: "All the missing Life Sciences articles part 2", General Discourse) Glennon RA, Ismaiel AE, Martin B, Poff D, Sutton M A preliminary behavioral investigation of PMMA, the 4-methoxy analog of methamphetamine Pharmacol. Biochem. Behav., 1988, 31(1), 9-13 Medline (PMID=3252264) Post 512563 (7is: "All the missing PBB articles part 4", General Discourse) Glennon RA, Yousif M, Patrick G Stimulus properties of 1-(3,4-methylenedioxyphenyl)-2-aminopropane (MDA) analogs Pharmacol. Biochem. Behav., 1988, 29(3), 443-449 Medline (PMID=2896360) Post 512563 (7is: "All the missing PBB articles part 4", General Discourse) Rosecrans JA, Glennon RA The effect of MDA and MDMA ("Ecstasy") isomers in combination with pirenpirone on operant responding in mice Pharmacol. Biochem. Behav., 1987, 28(1), 39-42 Medline (PMID=2889221) Post 512563 (7is: "All the missing PBB articles part 4", General Discourse) Glennon RA, Yousif M, Naiman N, Kalix P Methcathinone: a new and potent amphetamine-like agent Pharmacol. Biochem. Behav., 1987, 26(3), 547-551 Medline (PMID=3575369) Post 512563 (7is: "All the missing PBB articles part 4", General Discourse) Glennon RA, Little PJ, Rosecrans JA, Yousif M The effect of MDMA ("Ecstasy") and its optical isomers on schedule-controlled responding in mice Pharmacol. Biochem. Behav., 1987, 26(2), 425-426 Medline (PMID=2883666) Post 512563 (7is: "All the missing PBB articles part 4", General Discourse) Kalix P, Glennon RA Further evidence for an amphetamine-like mechanism of action of the alkaloid cathinone Biochem Pharmacol., 1986, 35(18), 3015-3019 Medline (PMID=3753515) Young R, Glennon RA Discriminative stimulus properties of amphetamine and structurally related phenalkylamines Med. Res. Rev., 1986, 6(1), 99-130 Medline (PMID=3512936) Lyon RA, Glennon RA, Titeler M 3,4-Methylenedioxymethamphetamine (MDMA): stereoselective interactions at brain 5-HT1 and 5-HT2 receptors Psychopharm. (Berl)., 1986, 88(4), 525-526 Medline (PMID=2871581) Schechter MD, Glennon RA Cathinone, cocaine and methamphetamine: similarity of behavioral effects Pharmacol. Biochem. Behav., 1985, 22(6), 913-916 Medline (PMID=4023025) Post 512563 (7is: "All the missing PBB articles part 4", General Discourse) Glennon RA, Young R, Hauck AE, McKenney JD Structure-activity studies on amphetamine analogs using drug discrimination methodology Pharmacol. Biochem. Behav., 1984, 21(6), 895-901 Medline (PMID=6522418) Post 496940 (lugh: "Glennon's article", Serious Chemistry) Glennon RA, Schechter MD, Rosecrans JA Discriminative stimulus properties of S(-)- and R(+)-cathinone, (+)-cathine and several structural modifications Pharmacol. Biochem. Behav., 1984, 21(1), 1-3 Medline (PMID=6463083) Post 512563 (7is: "All the missing PBB articles part 4", General Discourse) Aceto MD, Rosecrans JA, Young R, Glennon RA Similarity between (+)-amphetamine and amfonelic acid Pharmacol. Biochem. Behav., 1984, 20(4), 635-637 Medline (PMID=6728880) Post 512563 (7is: "All the missing PBB articles part 4", General Discourse) Glennon RA, Young R Further investigation of the discriminative stimulus properties of MDA Pharmacol. Biochem. Behav., 1984, 20(4), 501-505 Medline (PMID=6728867) Post 512565 (7is: "All the missing PBB articles part 5", General Discourse) Glennon RA, Young R MDA: an agent that produces stimulus effects similar to those of 3,4-DMA, LSD and cocaine Eur. J. Pharmacol., 1984, 99(2-3), 249-250 Medline (PMID=6145599) Schechter MD, Rosecrans JA, Glennon RA Comparison of behavioral effects of cathinone, amphetamine and apomorphine Pharmacol. Biochem. Behav., 1984, 20(2), 181-184 Medline (PMID=6718445) Post 512565 (7is: "All the missing PBB articles part 5", General Discourse) Glennon RA, Young R MDA: a psychoactive agent with dual stimulus effects Life Sci., 1984, 34(4), 379-383 Medline (PMID=6694526) Post 508287 (not existing) Glennon RA, Young R, Soine W 1-(2,3-Methylenedioxyphenyl)-2-aminopropane (2,3-MDA): a preliminary investigation Gen. Pharmacol., 1984, 15(4), 361-362 Medline (PMID=6149169) Glennon RA, Young R, Rosecrans JA, Anderson GM Discriminative stimulus properties of MDA analogs Biol. Psychiatry, 1982, 17(7), 807-814 Medline (PMID=6126227) Glennon RA, Liebowitz SM Serotonin receptor affinity of cathinone and related analogues J. Med. Chem., 1982, 25(4), 393-397 Medline (PMID=7069716) Glennon, R. A.; Showalter, D The Effects of Cathinone and Several Related Derivatives on Locomotor Activity Res. Commun. Subst. Abuse 1981, 2, 186 No PubMed entry or DOI found Kalix, P.; Yousif, M. Y.; Glennon, R. A Differential effect of the enantiomers of methylenedioxyamphetamine (MDMA) on the release of radioactivity from [3H]dopamine-prelabeled rat striatum Res. Commun. Substance Abuse 1988, 9, 45-51 No PubMed entry or DOI found Glennon, R. A.; Misenheimer, B Stimulus effects of N-mono ethyl-(3,4-methylenedioxyphenyl)-2-aminopropane (MDE) and N-hydroxy-1-(3,4-methylenedioxyphenyl)-2-aminopropane (N-OH MDA) in rats trained to discriminate MDMA from saline Pharmacol. Biochem. Behav., 1989, 33, 900-912 No PubMed entry or DOI found Dal Cason, T.; Young, R.; Glennon, R. A Cathinone: An investigation of several N-alkyl and methylenedioxy-substituted analogs Pharmacol. Biochem. Behav., 1997, 58, 1109-1116 No PubMed entry or DOI found Young, R.; Gabryszuk, M.; Glennon, R. A (-)Ephedrine and caffeine mutually potentiate one anothers amphetamine-like stimulus effects Pharmacol. Biochem. Behav., 1998, 61, 169-173 No PubMed entry or DOI found Young, R.: Glennon, R. A Discriminative stimulus properties of (-)ephedrine Pharmacol. Biochem. Behav., 1998, 60, 771-775 No PubMed entry or DOI found Glennon, R. A.; Young, R (+)Amphetamine stimulus generalization to an herbal ephedrine product Pharmacol. Biochem. Behav., 2000, 65, 655-658 No PubMed entry or DOI found Malmusi, L.; Dukat, M.; Young, R.; Teitler, M.; Darmani, N.; Ahmad, B.; Smith, C.; Glennon, R. A 1,2,3,4- Tetrahydroisoquinolines and related analogs of the phenylalkylamine designer drug MDMA Med. Chem. Res., 1996, 6, 412-426 No PubMed entry or DOI found The sigma receptor Ablordeppey SY, Fischer JB, Law H, Glennon RA Probing the proposed phenyl-A region of the sigma-1 receptor Bioorg. Med. Chem., 2002, 10(8), 2759-2265 Medline (PMID=12057665) Ablordeppey SY, Fischer JB, Glennon RA Is a nitrogen atom an important pharmacophoric element in sigma ligand binding? Bioorg. Med. Chem., 2000, 8(8), 2105-2111 Medline (PMID=11003156) Glennon RA, Ablordeppey SY, Ismaiel AM, el-Ashmawy MB, Fischer JB, Howie KB Structural features important for sigma 1 receptor binding J. Med. Chem., 1994, 37(8), 1214-1219 Medline (PMID=8164264) Glennon RA, Yousif MY, Ismaiel AM, el-Ashmawy MB, Herndon JL, Fischer JB, Server AC, Howie KJ Novel 1-phenylpiperazine and 4-phenylpiperidine derivatives as high-affinity sigma ligands J. Med. Chem., 1991, 34(12), 3360-3365 Medline (PMID=1662725) Glennon RA, Ismaiel AM, Smith JD, Yousif M, el-Ashmawy M, Herndon JL, Fischer JB, Howie KJ, Server AC Binding of substituted and conformationally restricted derivatives of N-(3-phenyl-n-propyl)-1-phenyl-2-aminopropane at sigma-receptors J. Med. Chem., 1991, 34(6), 1855-1859 Medline (PMID=1648139) Glennon RA, Smith JD, Ismaiel AM, el-Ashmawy M, Battaglia G, Fischer JB Identification and exploitation of the sigma-opiate pharmacophore J. Med. Chem., 1991, 34(3), 1094-1098 Medline (PMID=1848295) Glennon RA, Battaglia G, Smith JD (-)PPAP: a new and selective ligand for sigma binding sites Pharmacol. Biochem. Behav., 1990, 37(3), 557-559 Medline (PMID=1965044) Post 512565 (7is: "All the missing PBB articles part 5", General Discourse) Glennon, R.A., El-Ashmawy, M., Fischer, J.B., Burke Howie, K.J., Ismaiel, A.M N-Substituted 5-phenyl pentylamines: A new class of s receptor ligands Med. Chem. Res., 1991, 1, 207-212 No PubMed entry or DOI found Ablordeppey, S.Y.; El-Ashmawy, M. B.; Glennon, R.A Analysis of the structure-activity relationships of sigma receptor ligands Med. Chem. Res. 1991, 1, 425-438 No PubMed entry or DOI found El-Ashmawy, M.; Ablordeppey, S.Y.; Issa, H.; Gad, L.; Fischer, J.B.; Burke Howie, K. J.; Glennon, R. A Further investigation of 5-phenylpentylamine derivatives as novel s receptor ligands Med. Chem. Res., 1992, 2, 119-126 No PubMed entry or DOI found Ablordeppey, S.Y.; El-Ashmawy, M. B.; Glennon, R.A Analysis of the structure-activity relationships of sigma receptor ligands Med. Chem. Res., 1992, 2, 425-438 No PubMed entry or DOI found Ablordeppey, S.Y.; Fischer, J.B.; Burke Howie, K.J.; Glennon, R.A Design, synthesis and binding of sigma receptor ligands derived from butaclamol Med. Chem. Res., 1992, 2, 368-375 No PubMed entry or DOI found Abou-Gharbia, M.; Ablordeppey, S.Y.; Glennon, R.A Sigma receptors and their ligands: The Sigma Enigma Ann. Rep. Med. Chem., 1993, 28, 1-10 No PubMed entry or DOI found Ablordeppey, SY; Ashmawy, M.; Fischer, J. B.; Glennon, R. A A CoMFA investigation of sigma receptor binding affinity: Reexamination of a spurious sigma ligand Eur. J. Med. Chem., 1998, 33, 625-633 No PubMed entry or DOI found Ablordeppey, SY; Issa, H; Fischer, JB; Burke Howie, KJ; Glennon, RA Synthesis and structure-affinity relationship studies of sigma ligands related to haloperidol Med. Chem. Res., 1993, 3, 131-138 No PubMed entry or DOI found Articles dealing with synthetic methods Glennon, R. A.; Bass, R. G.; Schubert, E Alkylation of thiazolo[3,2-a]pyrimidin-5,7-diones J. Heterocyclic Chem., 1979, 16, 903 No PubMed entry or DOI found Glennon, R. A.; Rogers, M. E.; El-Said, M. K Imidazo[1,2a]-pyrimidines and 1,2,4-triazolo[1,5-a]pyrimidines: Two new examples of mesoionic xanthine analogs J. Heterocyclic Chem., 1980, 17, 337 No PubMed entry or DOI found Glennon, R. A.; Schubert, E.; Bass, R. G Synthesis of Mesoionic Xanthine Nucleosides Tetrahedron Lett. 1981, 29, 2753 No PubMed entry or DOI found Salley, J. J.; Glennon, R. A Studies on Simplified Ergoline Derivatives. A General Six-step Synthesis of Phenyl- Substituted4-Methyl-3,4a,5,6,10b-hexahydrobenzo[f]quinolin-1(2H)-one Analogs J. Heterocyclic Chem., 1982, 19, 545 No PubMed entry or DOI found Schubert, E. M.; Bass, R. G.; Glennon, R. A Synthesis of mesoionic xanthine nucleosides Nucleosides/ Nucleotides, 1983, 2, 127 No PubMed entry or DOI found Mbagwu, G.; Bass, R. G.; Glennon, R. A Carbon-13 Nuclear Magnetic Resonance Spectra of some Mesoionic Xanthine Analogs Org. Magnetic Res., 1983, 21, 527 No PubMed entry or DOI found Glennon, R. A.; Tejani, S Mesoionic Nucleosides: Studies on Mesoionic Imidazo[2,1-b]-1,3-thiazine Derivatives Nucleosides/Nucleotides, 1984, 3, 389 No PubMed entry or DOI found Schubert, E. M.; Schram, K. H.; Glennon, R. A Mass spectrometry of modified nucleic acid bases and nucleosides. Class II mesoionic nucleosides and bases derived from thiazolo[3,2-a]pyrimidine-5,7-diones J. Heterocyclic. Chem., 1985, 22, 889 No PubMed entry or DOI found Mbagwu, G. O.; Bass, R. G.; Glennon, R. A Studies of amine-induced ring-opening of some mesoionic xanthines J. Heterocyclic Chem., 1985, 22, 465 No PubMed entry or DOI found Kerdawy, M.; Bayomi, S.; Shehata, I; Glennon, R. A Condensed 1,2,3-triazines: 1,3,4-thiadiazolo[3,2-a]-1,3, 5-triazines and isoxazolo[2,3-a]-1,3,5-triazines J. Heterocyclic Chem., 1987, 24, 501-504 No PubMed entry or DOI found Shehata, I.; Glennon, R. A Mesoionic isoxazolo[2,3-a]pyrimidindiones and 1,3,4-oxadiazolo[3,2-a]- pyrimidindiones as potential adenosine antagonists J. Heterocyclic Chem., 1987, 24, 1291-1295 No PubMed entry or DOI found Kerdawy, M. M.; Ismaiel, A. M.; Gineinah, M.; Glennon, R. A A convenient synthesis of 3-aryl-1,2,4-triazolo [4,3-c]quinazolines J. Heterocyclic Chem., 1990, 27, 497-501 No PubMed entry or DOI found Gineinah, M.; Ismaiel, A. M.; Kerdawy, M.; Glennon, R. A Mesoionic 1,2,4-triazolo[4,3-c]quinazolines J. Heterocyclic Chem., 1990, 27, 723-726 No PubMed entry or DOI found Coburn, R. A.; Carapellotti, R. A.; Glennon, R. A A PPP p-SCF variable integral study of mesoionic analogs based on six-membered ring mesoionic systems J. Heterocyclic Chem., 1973, 10, 479 No PubMed entry or DOI found Coburn, R. A.; Glennon, R. A Synthesis and properties of mesoionic thiazolo[3,2-a]pyrimidin-5,7-diones J. Heterocyclic Chem., 1973, 10, 487 No PubMed entry or DOI found Coburn, R. A.; Bhooshan, B.; Glennon, R. A The preparation of 2-alkylamino-1,3,4-thiadiazoles J. Org. Chem., 1973, 38, 3947 No PubMed entry or DOI found Glennon, R. A.; Von Strandtmann, M Cyclodehydration of N-heteroarylcarbamoylmethylbenzamides J. Heterocyclic Chem., 1975, 12, 135 No PubMed entry or DOI found The nicotinic acetyl choline receptor Glennon RA, Dukat M alpha4beta2 nACh receptor pharmacophore models Bioorg. Med. Chem. Lett., 2004, 14(8), 1841-1844 Medline (PMID=15050612) Glennon RA, Dukat M, Liao L Musings on alpha4beta2 nicotinic acetylcholine (nACh) receptor pharmacophore models Curr. Top. Med. Chem., 2004, 4(6), 631-644 Medline (PMID=14965299) Dogruer D, Lee M, Dukat M, Damaj MI, Martin BR, Glennon RA 3-(4-Aminobutyn-1-yl)pyridines: binding at alpha4beta2 nicotinic cholinergic receptors Bioorg. Med. Chem. Lett., 2004, 14(2), 523-526 Medline (PMID=14698195) Ferretti G, Dukat M, Giannella M, Piergentili A, Pigini M, Quaglia W, Damaj MI, Martin BR, Glennon RA Binding of nicotine and homoazanicotine analogues at neuronal nicotinic acetylcholinergic (nACh) receptors Bioorg. Med. Chem. Lett., 2003, 13(4), 733-735 Medline (PMID=12639569) Ferretti G, Dukat M, Giannella M, Piergentili A, Pigini M, Quaglia W, Damaj MI, Martin BR, Glennon RA Homoazanicotine: a structure-affinity study for nicotinic acetylcholine (nACh) receptor binding J. Med. Chem., 2002, 45(21), 4724-4731 Medline (PMID=12361399) Dukat M, El-Zahabi M, Ferretti G, Damaj MI, Martin BR, Young R, Glennon RA (-)6-n-Propylnicotine antagonizes the antinociceptive effects of (-)nicotine Bioorg. Med. Chem. Lett., 2002, 12(20), 3005-3007 Medline (PMID=12270194) Lee M, Dukat M, Liao L, Flammia D, Damaj MI, Martin B, Glennon RA A comparison of the binding of three series of nicotinic ligands Bioorg. Med. Chem. Lett., 2002, 12(15), 1989-1992 Medline (PMID=12113825) Young R, Glennon RA Nicotine and bupropion share a similar discriminative stimulus effect Eur. J. Pharmacol., 2002, 443(1-3), 113-118 Medline (PMID=12044800) Dukat M, Damaj IM, Young R, Vann R, Collins AC, Marks MJ, Martin BR, Glennon RA Functional diversity among 5-substituted nicotine analogs; in vitro and in vivo investigations Eur. J. Pharmacol., 2002, 435(2-3), 171-180 Medline (PMID=11821023) Ferretti G, Dukat M, Giannella M, Piergentili A, Pigini M, Quaglia W, Damaj MI, Martin BR, Glennon RA Chain-lengthened and imidazoline analogues of nicotine Bioorg. Med. Chem. Lett., 2000, 10(23), 2665-2668 Medline (PMID=11128647) Glennon RA, Dukat M Central nicotinic receptor ligands and pharmacophores Pharm. Acta Helv., 2000, 74(2-3), 103-114 Medline (PMID=10812946) Flammia D, Dukat M, Damaj MI, Martin B, Glennon RA Lobeline: structure-affinity investigation of nicotinic acetylcholinergic receptor binding J. Med. Chem., 1999, 42(18), 3726-3731 Medline (PMID=10479304) Damaj MI, Fei-Yin M, Dukat M, Glassco W, Glennon RA, Martin BR Antinociceptive responses to nicotinic acetylcholine receptor ligands after systemic and intrathecal administration in mice J. Pharmacol. Exp. Ther., 1998, 284(3), 1058-1065 Medline (PMID=9495867) Glennon, R.A.; Maarouf, R.; Fahmy, S.; Martin, B.; Fan, F.; Yousif, M.; Shafik, R.; Dukat, M Structure-affinity relationships of simple nicotine analogs Med. Chem. Res., 1993, 2, 546-551 No PubMed entry or DOI found Dukat, M.; Damaj, M. I.; Glassco, W.; Dumas, D.; May, E. L.; Martin, B. R.; Glennon, R. A Epibatidine: A very high affinity nicotine-receptor ligand Med. Chem. Res., 1994, 4, 131-139 No PubMed entry or DOI found Glennon, R.A.; Herndon, J.; Dukat, M Epibatidine-aided studies toward definition of a nicotine receptor pharmacophore Med. Chem. Res., 1994, 4, 461-473 No PubMed entry or DOI found Glennon, R.A.; Fiedler, W.; Dukat, M.; Damaj, I.; Martin, B Pyrrolidine-modified analogues of nicotine: a structure-affinity investigation Eur. J. Med. Chem., 1996, 31, 875-888 No PubMed entry or DOI found Glennon, R. A.; Dukat, M Nicotine receptor ligands Med. Chem. Res., 1996, 6, 465-486 No PubMed entry or DOI found Damaj, M. I.; Glassco, W.; Dukat, M.; May, E. L.; Glennon, R. A.; Martin, B. R Pharmacology of novel nicotinic analogs Drug Dev. Res., 1996, 38, 177-187 No PubMed entry or DOI found Dukat, M.; Dowd, M.; Damaj, M. I.; Martin, B.; El-Zahabi, M. A.; Glennon, R. A Synthesis, receptor binding, and QSAR studies on 6-subtituted nicotine derivatives as cholinergic ligands Eur. J. Med. Chem., 1999, 34, 31-40 No PubMed entry or DOI found Cheng, Y.-X.; Dukat, M.; Dowd, M.; Fiedler, W.; Martin, B.; Damaj, M. I.; Glennon, R. A Synthesis and binding of 6,7,8,9-tetrahydro-5H-pyrido[3,4-d]azepine and related ring-opened analogs at central nicotinic receptors Eur. J. Med. Chem., 1999, 34, 177-190 No PubMed entry or DOI found Dukat M, Glennon RA Epibatidine: impact on nicotinic receptor research Cell. Mol. Neurobiol., 2003, 23(3), 365-378 Medline (PMID=12825833) The imidazoline receptor Tyacke RJ, Lau A, Grella B, Glennon RA, Nutt DJ, Hudson AL Investigation of the affinities of two new beta-carbolines for rat brain imidazoline(2) receptors Ann N Y Acad Sci., 2003, 1009, 361-363 Medline (PMID=15028612) Chang-Fong J, Tyacke RJ, Lau A, Westaway J, Hudson AL, Glennon RA Pyrazino[1,2-a]indoles as novel high-affinity and selective imidazoline I(2) receptor ligands Bioorg. Med. Chem. Lett., 2004, 14(4), 1003-1005 Medline (PMID=15013010) Glennon RA, Grella B, Tyacke RJ, Lau A, Westaway J, Hudson AL Binding of beta-carbolines at imidazoline I2 receptors: a structure-affinity investigation Bioorg. Med. Chem. Lett., 2004, 14(4), 999-1002 Medline (PMID=15013009) Glennon RA, Grella B, Tyacke RJ, Lau A, Westaway J, Hudson AL Binding of an imidazopyridoindole at imidazoline I2 receptors Bioorg. Med. Chem. Lett., 2004, 14(2), 527-529 Medline (PMID=14698196) Husbands SM, Glennon RA, Gorgerat S, Gough R, Tyacke R, Crosby J, Nutt DJ, Lewis JW, Hudson AL beta-carboline binding to imidazoline receptors Drug Alcohol Depend., 2001, 64(2), 203-208 Medline (PMID=11543990) Post 494854 (Nicodem: "Papers on beta-carbolines", General Discourse) Articles on various subjects Dukat M, Taroua M, Dahdouh A, Siripurapu U, Damaj MI, Martin BR, Glennon RA (+/-)8-Amino-5,6,7,8-tetrahydroisoquinolines as novel antinociceptive agents Bioorg. Med. Chem. Lett., 2004, 14(14), 3651-3654 Medline (PMID=15203136) Glennon RA, Ismaiel AM, Ablordeppey S, El-Ashmawy M, Fisher JB Thioxanthene-derived analogs as [Formula: see text] receptor ligands Bioorg. Med. Chem. Lett., 2004, 14(9), 2217-2220 Medline (PMID=15081012) Post 508287 (not existing) Glennon RA [In Process Citation] Prog. Med. Chem., 2004, 42, 55-123 Medline (PMID=15003719) Simsek R, Chang-Fong J, Lee M, Dukat M, Imad Damaj M, Martin BR, Glennon RA Quaternary ammonium 3-(aminoethoxy)pyridines as antinociceptive agents Bioorg. Med. Chem. Lett., 2003, 13(17), 2917-2920 Medline (PMID=14611857) Bondarev ML, Bondareva TS, Young R, Glennon RA Behavioral and biochemical investigations of bupropion metabolites Eur. J. Pharmacol., 2003, 474(1), 85-93 Medline (PMID=12909199) Glennon RA, Young R, Rangisetty JB Further characterization of the stimulus properties of 5,6,7,8-tetrahydro-1,3-dioxolo[4,5-g]isoquinoline Pharmacol. Biochem. Behav., 2002, 72(1-2), 379-387 Medline (PMID=11900809) https://www.rhodium.ws/pdf/glennon.2002.tdiq.pdf Hellberg M, Stubbins JF, Glennon RA A preliminary investigation of mesoionic xanthine analogues as inhibitors of platelet aggregation Bioorg. Med. Chem., 2000, 8(8), 1917-1923 Medline (PMID=11003136) Glennon RA, Dukat M, Westkaemper RB, Ismaiel AM, Izzarelli DG, Parker EM The binding of propranolol at 5-hydroxytryptamine1D beta T355N mutant receptors may involve formation of two hydrogen bonds to asparagine Mol. Pharmacol., 1996, 49(1), 198-206 Medline (PMID=8569707) Damaj MI, Glennon RA, Martin BR Involvement of the serotonergic system in the hypoactive and antinociceptive effects of nicotine in mice Brain Res. Bull., 1994, 33(2), 199-203 Medline (PMID=8275340) Glennon RA, Young R, Herndon JL Antagonism of a (+)N-allylnormetazocine stimulus by (-)PPAP and several structurally related analogs Pharmacol. Biochem. Behav., 1993, 45(4), 865-869 Medline (PMID=8105490) Post 512565 (7is: "All the missing PBB articles part 5", General Discourse) Young R, Glennon RA Zacopride and its optical isomers produce stereoselective antagonism of a 2-methylserotonin discriminative stimulus Eur. J. Pharmacol., 1992, 212(1), 117-119 Medline (PMID=1555633) Glennon RA, De Vry J, Spencer DG Jr, Glaser T Stimulus properties of tiflucarbine: a novel antidepressant agent Pharmacol. Biochem. Behav., 1990, 37(4), 769-771 Medline (PMID=2151199) Post 512565 (7is: "All the missing PBB articles part 5", General Discourse) Glennon RA, Pierson ME, McKenney JD Stimulus generalization of 1-(3-trifluoromethylphenyl)piperazine (TFMPP) to propranolol, pindolol, and mesulergine Pharmacol. Biochem. Behav., 1988, 29(1), 197-199 Medline (PMID=2895480) Post 512565 (7is: "All the missing PBB articles part 5", General Discourse) Young R, Glennon RA Stimulus properties of benzodiazepines: correlations with binding affinities, therapeutic potency, and structure activity relationships (SAR) Psychopharm. (Berl)., 1987, 93(4), 529-533 Medline (PMID=2893418) Young R, Glennon RA, Dewey WL Effects of pyrazolopyridines and a triazolopyridazine on the pentobarbital discriminative stimulus Psychopharm. (Berl)., 1987, 93(4), 494-497 Medline (PMID=2893416) Young R, Glennon RA, Brase DA, Dewey WL Potencies of diazepam metabolites in rats trained to discriminate diazepam Life Sci., 1986, 39(1), 17-20 Medline (PMID=3088348) Glennon RA, Tejani-Butt SM, Padgett W, Daly JW Mesoionic xanthine analogues: antagonists of adenosine receptors J. Med. Chem., 1984, 27(10), 1364-1367 Medline (PMID=6090665) Young R, Glennon RA, Dewey WL Stereoselective stimulus effects of 3-methylflunitrazepam and pentobarbital Life Sci., 1984, 34(20), 1977-1983 Medline (PMID=6328149) Post 508287 (not existing) Lund MQ, Kier LB, Glennon RA, Egle JL Jr Preliminary studies of mesoionic 3-(substituted-aryl)-psi-oxatriazoles as potential antihypertensive agents J. Med. Chem., 1982, 25(12), 1503-1505 Medline (PMID=7154013) Rogers ME, Glennon RA, Smith JD, Boots MR, Nanavati N, Maconaughey E, Aub D, Thomas S, Bass RG, Mbagwu G Mesoionic purinone analogues as inhibitors of cyclic-AMP phosphodiesterase: a comparison of several ring systems J. Med. Chem., 1981, 24(11), 1284-1287 Medline (PMID=6273558) Glennon RA, Salley JJ Jr, Steinsland OS, Nelson S Synthesis and evaluation of novel alkylpiperazines as potential dopamine antagonists J. Med. Chem., 1981, 24(6), 678-683 Medline (PMID=7252977) Glennon RA, Gaines JJ, Rogers ME Benz-fused mesoionic xanthine analogues as inhibitors of cyclic-AMP phosphodiesterase J. Med. Chem., 1981, 24(6), 766-769 Medline (PMID=6265639) Glennon RA, Rogers ME, Smith JD, El-Said MK, Egle JL Mesoionic xanthine analogues: phosphodiesterase inhibitory and hypotensive activity J. Med. Chem., 1981, 24(6), 658-661 Medline (PMID=6265635) Glennon RA, Schubert E, Jacyno JM, Rosecrans JA Studies on several 7-substituted N,N-dimethyltryptamines J. Med. Chem. 1980, 23(11), 1222-1226 Medline (PMID=6779006) https://www.rhodium.ws/pdf/7-substituted.dmt.pdf Rosecrans JA, Glennon RA Drug-induced cues in studying mechanisms of drug action Neuropharmacology. 1979, 18(12), 981-989 Medline (PMID=530379) Glennon RA, Rogers ME, Bass RG, Ryan SB Mesoionic xanthine analogs as inhibitors of cyclic AMP phosphodiesterase J. Pharm. Sci., 1978, 67(12), 1762-1765 Medline (PMID=214541) Coburn RA, Glennon RA Mesoionic purinone analogs. 7. In vitro antibacterial activity of mesoionic 1,3,4-thiadiazolo(3,2-a)pyrimidine-5,7-diones J. Med. Chem., 1974, 17(9), 1025-1027 Medline (PMID=4213245) Coburn RA, Glennon RA Mesoionic purinone analogs. IV. Synthesis and in vitro antibacterial properties of mesoionic thiazolo(3,2-a)pyrimidin-5,7-diones and mesoionic 1,3,4-thiadizolo(3,2-a)pyrimidin-5,7-diones J. Pharm. Sci., 1973, 62(11), 1785-1789 Medline (PMID=4202220) Watson, H.; Glennon, R.A Common drug interactions Anesthesia Update, 1978, 6, 1 No PubMed entry or DOI found Young, R.; Glennon, R. A.; Brase, D.; Dewey, W. L Potencies of diazepam metabolites in generalizing to the diazepam discriminative stimulus Life Sci., 1985, 39, 17 No PubMed entry or DOI found The tendency is to push it as far as you can |
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