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    Digest: Archive of "Wanted References" Volume 1   Please login to post  

(Chief Bee)
03-19-04 16:46
No 436354
User Picture 
      Archive of "Wanted References" Volume 1     

The thread Post 217986 (Rhodium: "Wanted references", Novel Discourse) in this forum for requesting journal articles which are out of reach for yourself often becomes cluttered with posts after a while (so that it is hard to see which articles are still wanted and which has been retrieved), and as it is a waste to just delete the posts containing links to the retrieved articles (other bees than the actual requester may find them interesting), I will from now on collect these links in this separate digest (sorted according to who retrieved them) one week after they were first posted in Post 217986 (Rhodium: "Wanted references", Novel Discourse).

This Digest only covers articles posted in March 2004 or earlier. For articles posted in April 2004 or later, please refer to Post 499541 (Rhodium: "Archive of "Wanted References" Volume 2", Novel Discourse)

Please PM me if any of the links below expire, so that I can remove them from this list.

Retrieved by Chimimanie:

For Lego: (copy and paste them because the link dont work):
Synthesis of psilocine from N, N-dimethyltryptamine
Comptes Rendus des Seances de l'Academie des Sciences, Serie C:  Sciences Chimiques  (1969),  269(1),  51-3

For Kinetic:

For Rhodium:
2,5-Dimethoxyallylbenzene isomerization with PdCl2(MeCN)2
Aust. J. Chem. 43, 777-781 (1990)

Synthesis of Methadone
Bull. Soc. Chim. Belg. 90(9), 977-82 (1981)

For Vitus_Verdegast:
5-iodo-2-aminoindan, a non-neurotoxic analogue of p-iodo-amphetamine
Nichols, D.E.; Johnson, M.P. and Oberlender, P.
Pharmacol. Biochem. Behav. 38, 1, p.135 (1991) (

And BTW Here is the ref requested by Dr Shulgin in TiHKAL #30:
Salutations Mr Shulginsmile

Retrieved by Rhodium:

For roger2003:
Zur Kenntnis der Glyoxylsäure
Hans Meyer
Chem. Ber. 34, 3593-93 (1904) (

For pHarmacist:
Deveral Derivatives of p-Chlorophenoxyacetic Acid
N. A. Zakharova, et al.
Chemical Abstracts, Vol 63, 17948 (1965) (
(Unfortunately I believe that you will have to make do with only the abstract - Rumor says that odd journal is only kept in a total of five libraries in the western world...)

For Merbst:
Synthesis and Biological Evaluation of 14-Alkoxymorphinans. 8. 14-Methoxymetopon, an Extremely Potent Opioid Agonist
H. Schmidhammer, A. Schratz, J. Mitterdorfer
Helv. Chim. Acta.  73, 1784-87 (1990) (

For Lego:
S-Oxidation products of alkylthioamphetamines
Rezende, Marcos Caroli; Nunez, Christian; Sepulveda-Boza, Silvia; Cassels, Bruce K.; Hurtado-Guzman, Claudio.
Synthetic Communications 32(17), 2741-2750 (2002) (

Bromodecarbonylation and Bromodecarboxylation of Electron-Rich Benzaldehydes and Benzoic Acids with Oxone® and Sodium Bromide
Bon-Suk Koo; Eun-Hoo Kim; Kee-Jung Lee
Synthetic Communications 32(15), 2275-2286 (2002) (

Alkylation of alkyl nitroacetates under PTC conditions    
Gogte, V. N.; Natu, A. A.; Pore, V. S.
Synthetic Communications 17(12),  1421-9 (1987) (
Abstract: Treatment of O2NCHRCO2R1 (I; R = H, R1 = Me; R = Me, R1 = Et) with p-R2C6H4CH2Br (R2 = H, Cl, MeO) and KHCO3 in DMF contg. TEBA gave 70-78% p-R2C6H4CH2CR(NO2)CO2R1.  Similar treatment of I (R = H, R1 = Me) with p-O2NC6H4CH2Br gave (p-NO2C6H4CH2)2C(NO2)CO2Me.

In situ reagents for thionation of amides, peptides and lactams
Dennis Brillon
Synthetic Communications 20(19), 3085-3095 (1990) (
Abstract: An agent, prepd. from 1:1 P2S5 and Na2CO3 in situ, is used for thionation of amides, amino acids, peptides, and lactams.  Yields range from 28 to 96%.
As mentioned in: Post 468717 (Lego: "Amide to thioamide to amine", Serious Chemistry)

For Aurelius:
Direct Conversions of Ethers to Esters by Trichloroisocyanuric Acid
Tet. Lett. 55, 5819-5820 (1968) (

The Oxidation of Alcohols and Ethers Using Calcium Hypochlorite [ Ca(OCl)2 ]
Tet. Lett. 23(1), 35-38 (1982) (

Oxidation Studies of Symmetrical and Unsymmetriclal Ethers - Comparison of Trichloroisocyanuric Acid and Hypochlorous Acid
Tetrahedron 27, 2671-2674 (1971) (

Allylbenzenes by Friedel-Craft alkylation with Allyl Alcohol, catalyzed by K-10 Acidic Clay
J. Chem. Soc. Perkin Trans 1, 3519-3520 (1994) (

For Twodogs:
J. Chem. Educ. 76, 1717 (1999) (

For Vitus_Verdegast:
Org. Proc. Res. Dev. 4, 534-543 (2000) (
(And if you look around you will find sections of this already posted here)

For Antoncho:
Haworth and Lapworth, J. Chem. Soc., 121, 76 (1922) (

For Captain_Mission:
Direct conversion of Bromohydrins to ketones by a free radical elimination of HBr
J. Org. Chem. Vol. 67(1), 312-313(2002) (

Simple, inexpensive procedure for the large-scale production of alkyl quinones
J. Org. Chem.; 1983; 48(17); 2932-2933. (

For Ganesha:
Amphetamine Analogs. II. Methylated Phenethylamines (Added 03-15-04):
Beng T. Ho, et. al.
J. Med. Chem. 13, 134-135 (1970) (

Psychotropic Phenylisopropylamines derived from Apiole and Dillapiole (Added 03-15-04):
Alexander T. Shulgin
Nature 215, 1494-95 (1967) (

Structure-Activity Relationships of One-Ring Psychotomimetics (Added 03-15-04):
Alexander T. Shulgin, Thornton Sargent, Claudio Naranjo
Nature 221, 537-541 (1969) (

For Chimimanie:
The Alkaloids, Vol III:

Acta Pharm. Suecia 16, 267-270 (1979) (Under the heading "A Novel Route for the Synthesis of Mescaline")

The use of nitrilium salts in the synthesis of heterocyclic compounds. I. Derivatives of 3,4-dihydroisoquinoline
Lora-Tamayo, Manuel; Madronero, Ramon; Munoz, Guillermo Garcia
Chem. Ber. 93, 289-297 (1960) (

The Preparation of Alkyl Chlorides
James F. Norris, Hazel B. Taylor
J. Am. Chem. Soc. 46(3), 753-757 (1924) (

Phenylalkylamines with potential psychotherapeutic utility.  2.  Nuclear substituted 2-amino-1-phenylbutanes.
Standridge, Robert T.; Howell, Henry G.; Tilson, Hugh A.; Chamberlain, John H.; Holava, Henry M.; Gylys, Jonas A.; Partyka, Richard A.; Shulgin, Alexander T. 
Journal of Medicinal Chemistry  (1980),  23(2),  154-62. (

Synthesis and body distribution of several iodine-131-labeled central nervous system active drugs.
Braun, Ulrich; Shulgin, Alexander T.; Braun, Gisela; Sargent, Thornton, III.
Journal of Medicinal Chemistry  (1977),  20(12),  1543-6. (

1-[4-(3-Phenylalkyl)phenyl]-2-aminopropanes as 5-HT2A Partial Agonists
Cynthia S. Dowd, Katharine Herrick-Davis, Christina Egan, Ann DuPre, Carol Smith, Milt Teitler, and Richard A. Glennon
J. Med. Chem. 43(16) pp 3074 - 3084 (2000) (

Iodine-125 labeled 1-(2,5-dimethoxy-4-iodophenyl)-2-aminopropane: an iodinated radioligand that specifically labels the agonist high-affinity state of 5-HT2 serotonin receptors
Richard A. Glennon, Mark R. Seggel, William H. Soine, Katherine Herrick-Davis, Robert A. Lyon, Milt Titeler
J. Med. Chem. 31(1), 5-7 (1988) (

Phenylalkylamines with potential psychotherapeutic utility. 1. 2-Amino-1-(2,5-dimethoxy-4-methylphenyl)butane
Robert T. Standridge, Henry G. Howell, Jonas A. Gylys, Richard A. Partyka, Alexander T. Shulgin
J. Med. Chem. 19(12), 1400-1404 (1976) (

Phenylalkylamines with potential psychotherapeutic utility. 2. Nuclear substituted 2-amino-1-phenylbutanes
Robert T. Standridge, Henry G. Howell, Hugh A. Tilson, John H. Chamberlain, Henry M. Holava, Jonas A. Gylys, Richard A. Partyka, Alexander T. Shulgin
J. Med. Chem. 23(2), 154-162 (1980) (

Potential psychotomimetics.  New bromoalkoxyamphetamines
Sepulveda, Silvia; Valenzuela, Ricardo; Cassels, Bruce K.
Journal of Medicinal Chemistry 15(4), 413-15 (1972) (

Cross-linking and sequence-specific alkylation of DNA by aziridinylquinones. 3. Effects of alkyl substituents.
Hargreaves, Robert H. J.; O'Hare, C. Caroline; Hartley, John A.; Ross, David; Butler, John.   
Journal of Medicinal Chemistry  (1999),  42(12),  2245-2250. (

Isomeric cyclopropyl ring-methylated homologs of trans-2-(2,5-dimethoxy-4-methylphenyl)cyclopropylamine, an hallucinogen analog.
Jacob, James N.; Nichols, David E.   
Journal of Medicinal Chemistry  (1982),  25(5),  526-30. (

The article below is very interesting, as it contains novel routes to phenyl-2-propanones and other fun stuff.

2,4-Diaminothieno[2,3-d]pyrimidine analogs of trimetrexate and piritrexim as potential inhibitors of Pneumocystis carinii and Toxoplasma gondii dihydrofolate reductase.
Rosowsky, Andre; Mota, Clara E.; Wright, Joel E.; Freisheim, James H.; Heusner, James J.; McCormack, John J.; Queener, Sherry F.
Journal of Medicinal Chemistry 36, 3103-12 (1993) (

For Tdurden969:
Electrosynthesis attempts of tetrahydridoborates
E. L. Gyenge & C. W. Oloman
Journal of Applied Electrochemistry 28(10), 1147-1151 (1998) (

A new approach to electrochemical production of benzaldehyde from toluene in an undivided cell in the presence of the couple V5+/V4+
Qingfeng Y.,  Xiaoping L., Xiuling Z.
Journal of Applied Electrochemistry 33(3/4), 273-277 (2003) (

A study on wastewater minimization in indirect electrochemical synthesis of benzaldehyde
Ding Zhoua, Zhirong Suna and Wanli Hu
Water Science and Technology 34(10), 113-120 (1996) (

For fallen_angel:
Friedel-Crafts and Related Reactions. Chapter 37, Section I-II: Alkene Acylation
C.D. Nenitzescu & A.T. Balaban
Volume III, Part 2, pp. 1032-1066 (

Friedel-Crafts and Related Reactions. Chapter 37: References
C.D. Nenitzescu & A.T. Balaban
Volume III, Part 2, pp. 1136-1152 (

A Convenient Preparation of Tetrahydro-4H-pyran-2-one
G. R. Owen & C. B. Reese
J. Chem. Soc. C, 2401-2403 (1970) (

For Java:
Chemistry of nitrogen radicals. VI. The free-radical addition of dialkyl-N-chloramines to substituted olefins
J. Org. Chem.; 1967; 32(11); 3273-3284. (

Nonaromatic aminium radicals
Chem. Rev.; 1978; 78(3); 243-274. (

Radical addition of protonated N-chloroamines to olefins
Tet. Lett. 3163-3166 (1966) (

Synthesis of Arylpropylamines. I. From Allyl Chloride
T. M. Patrick, Jr., E. T. McBee, H. B. Hass;
J. Am. Chem. Soc.; 1946; 68(6); 1009-1011. (

Synthesis of allylic amines through the palladium-catalyzed hydroamination of allenes
Tetrahedron Letters 36(22), 3857-3860 (1995) (

Preparation of Aldehydes from Alkenes by the Addition of Carbon Monoxide and Hydrogen with Cobalt Carbonyls as Intermediates
Homer Adkins, George Krsek
J. Am. Chem. Soc. 70, 383-386 (1948) (

Über die Beziehungen zwischen dem assym. Methyl-phenyl-äthylen-glycol und den ihm entsprechenden Anhydro-Formen
S. Danilow & E. Venus-Danilowa
Chem. Ber. 60, 1050-1069 (1927) (

Chem. Ber. 89, 2641-2644 (1956) (

Arylation of several carbanions by the SRN1 mechanism
Roberto A. Rossi, J. F. Bunnett;
J. Org. Chem.; 1973; 38(17); 3020-3025. (

SRN1 phenylation of nitrile carbanions and ensuing reactions. New route to alkylbenzenes
J. F. Bunnett, Bernhard F. Gloor;
J. Org. Chem.; 1973; 38(24); 4156-4163. (

Mesitylation and phenylation of picolyl anions by the SRN1 mechanism
J. F. Bunnett, Bernhard F. Gloor;
J. Org. Chem.; 1974; 39(3); 382-384. (

Palladium-catalyzed arylation of siloxycyclopropanes with aryl triflates. Carbon chain elongation via catalytic carbon-carbon bond cleavage
Satoshi Aoki, Tsutomu Fujimura, Eiichi Nakamura, Isao Kuwajima
J. Am. Chem. Soc. 110, 3296-3298 (1988) (
Ferrous ion catalysis of reactions of nucleophiles with aryl halides
Carlo Galli, J. F. Bunnett
J. Org. Chem. 49, 3041-3042 (1984) (

For anyone intrerested in the above arylations, I suggest that you take a look at the articles below:

Retrieved by ChemisTris:

For Rhodium:
Behavioral properties of psychoactive phenylisopropylamines in rats
European Journal of Pharmacology 76(4), 353-360 (1981) (

Synthesis of MDP2P
Synthetic Communications 24(2), 145 (1994) (

For Vitus_Verdegast:
Heterocycles 46, 91-94 (1997) (
J. Nat. Prod. 60(11), 1196-98 (1997) (

The Pharmacology and Clinical Pharmacology of 3,4-Methylenedioxymethamphetamine (MDMA, "Ecstasy")
A. Richard Green, Annis O. Mechan, J. Martin Elliott, Esther O'shea, M. Isabel Colado
Pharmacol. Rev., 5533-5600 (2003) (

Differences in potency and efficacy of a series of phenylisopropylamine/phenylethylamine pairs at 5-HT2A and 5-HT2C receptors
Claudio Acuña-Castillo, Claudio Villalobos, Pablo R. Moya, Patricio Sáez, Bruce K. Cassels, and J. Pablo Huidobro-Toro
British Journal of Pharmacology 136, 510-519 (2002) (

For pHarmacist:
Tetrahedron Letters 10(39), 3375-3376 (1969) (

Retrieved by FreakyDMT:

For Rhodium:
10% Pd/C and HCOOH transfer hydrogenolysis of common protection groups
Indian journal of chemistry. Section B, 41(5):1064-1067 (2002) (

Retrieved by Kinetic:

For Chimimanie:

Selective deprotection of esters using magnesium and methanol
Tet. Lett. 35(34), 6207-6210 (1994) (

Retrieved by Lego:

For Rhodium:
J Chem Res (Miniprint) 1137-1145 (1982)

For Chimimanie:
Phenylbutanoids from Zingiber cassumunar.    
Tuntiwachwuttikul, Pittaya; Pancharoen, Orasa; Jaipetch, Thaworn; Reutrakul, Vichai.   
Phytochemistry (Elsevier)  (1981),  20(5),  1164-5. (

Studies on Thai medicinal plants.  Part VIII.  Further characterization of the constituents of a Thai medicinal plant, Zingiber cassumunar Roxb.  
Kuroyanagi, Masanori; Fukushima, Seigo; Yoshihira, Kunitoshi; Natori, Shinsaku; Dechatiwongse, Thaweephol; Mihashi, Kunihide; Nishi, Masatoshi; Hara, Shuuji.    
Chemical & Pharmaceutical Bulletin  (1980),  28(10),  2948-59 (

Synthesis and hypolipidemic activity of modified side chain a-asarone homologues    
Cruz, Adriana; Garduno, Leticia; Salazar, Maria; Martinez, Elizdath; Jimenez-Vazquez, Hugo A.; Diaz, Francisco; Chamorro, German; Tamariz, Joaquin.
Arzneimittel-Forschung  (2001),  51(7),  535-544 (

For Vitus-Verdegast:
J. Pharm. Sci., 1967, 56, 970-973 ( (Added 02-15-04):
Trifluromethyl analogs of amphetamine and norephedrine
Roger M. Pinder, Alfred Burger

Arzneimittel-Forschung , 1970, 20, 245-246 ( (Added 02-15-04):
m- and p-Hydroxy-1-cyanophenethylamine
Roger M. Pinder, Alfred Burger, E. J. Ariens

For Azole
Synthesis of Concave Receptors Derived from Diphenylglycoluril. (Added 02-15-04):
Sijbesma, R. P.; Nolte, R. J. M.
Recl. Trav. Chim. Pays-Bas, 1993, 112, 643-647 (
Synthesis of 1,4-bis(2-chloroethoxy)benzene by PTC alkylation of hydroquinone (ref. #23 from Dihydrobenzofuran Analogues of Hallucinogens. 3. (

Retrieved by moo:

For Chimimanie:
Synthesis of compounds with potential central nervous system stimulant activity. I.
2-Amino-2-oxazolin-4-one-5-spirocycloalkanes and 2-amino-2-oxazolin-4-one-5-spiro(4'-piperidines)

Michael R. Harnden, Ray R. Rasmussen
J. Med. Chem. 12, 919-921 (1969) (

Synthesis of compounds with potential central nervous system stimulant activity. II.
5-Spiro-substituted 2-amino-2-oxazolines

Michael R. Harnden, Ray R. Rasmussen
J. Med. Chem. 13, 305-308 (1970) (

Synthesis and serotonin receptor affinities of a series of enantiomers of a-methyltryptamines:  evidence for the binding conformation of tryptamines at serotonin 5-HT1B receptors.
Nichols, David E.; Lloyd, David H.; Johnson, Michael P.; Hoffman, Andrew J.   
Journal of Medicinal Chemistry  (1988),  31(7),  1406-12. (

Retrieved by Java:

For Rhodium:
4-bromo-2,5-dimethoxyphenethylamine (2C-B): A review of the public domain literature.
Cole M.D,Lea C and Oxley N.
Science & Justice 42(4), 223-224 (2002) (

For ChemisTris:

New synthetic route for the preparation of potentially hypocholesterolemic analogs of alpha-asarone.
Determination of E/Z isomer content in natural and synthetic mixtures of alpha-asarone and its analogs.

Munoz, Heber; Diaz, Francisco; Sanchez, Adrian; Barajas, Marcelino; Labarrios, Fernando; Tamariz, Joaquin.   
Acta Mexicana de Ciencia y Tecnologia, 11(41), 51-62 (1993) (

Retrieved by 7is:

For Manichi:
Binding of Phenylalkylamine Derivatives at 5-HT1C and 5-HT2 Serotonin Receptors: Evidence for a Lack of Selectivity
Richard. A. Glennon
J. Med. Chem, 734 (1992) (

The Ethyl Homologs of 2,4,5-Trimethoxyphenylisopropylamines
Alexander T. Shulgin
J. Med. CHem 11, 196-187 (1968) (

For Rhodium:
Drug Discrimination and Receptor Binding Studies of N-Isopropyl Lysergamide Derivates
Huang, Marona-Lewicka, Pfaff, Nichols
Pharmacology, Biochmistry and Behavior 47(3), 667-673 (1994) (

Ergot Peptide Alkaloid Spectra of Claviceps-Infected Tall Fescue, Wheat, and Barley
James K. Porter, Charles W. Bacon, Ronald D. Plattner, and Richard F. Arrendale.
J. Agric. Food Chem. 35, 359-361 (1987) (

Synthesis of some fluorinated nitro-olefins
R. Jacobo, A. Cota, E. Rogel, J. D. Garcia, I. A. Rivero, L. H. Hellberg and R. Somanathan
Journal of Fluorine Chemistry, 67(3), 253-255 (1994) (

For Potter
Colour reactions of some aromatic ethers found in essential oils
Janet E. Forrest, R. Richard and R. A. Heacock
Journal of Chromatography A, 65(2), 439-444 (1972) (

For Vitus
Alfred Burger, Stuart E. Zimmerman, and E. J. Ariëns
J. Med. Chem. 9, 469 (1966) (

For Ganesha:
Forty years of hydride reductions latest addition (03-19-04):
Herbert C. Brown and S. Krishnamurthy
Tetrahedron 1979, 35, 567-607 (1979)

Retrieved by dioulasso:

For Rhodium:
Copper(II)-B-cyclodextrin aided oxidation of eugenol
Indian Journal Of Chemistry. Sect. B. 42(2), 369-371 (2003) (

Zinc/hydrazine: A low cost-facile system for the reduction of nitro compounds
Indian Journal Of Chemistry. Sect. B.  42(1), 180-183 (2003) (

Reduction of oximes with NaBH4/CuSO4/MeOH
Indian journal of chemistry. Section B,  41(5):1072-1074 (2002) (

Sodium Borohydride-Iodine, an Efficient Reagent for Reductive Amination of Aromatic Aldehydes
Ira Saxena, Ruli Borah, Jadab C. Sarma
Indian Journal of Chemistry Sect. B, 41(9), 1970-1971 (2002) (
(claimed to work only for benzaldehydes, not aliphatic carbonyl compounds)

For Vitus Verdegast:
Solvent-free Microwave Knoevenagel condensation catalyzed by NaCl or NH4OAc-AcOH
Indian Journal of Chemistry, Sect. B. 39(6), 403-405 (2000) (

Cobalt(II)Chloride Hexahydrate - Zinc - DMF - Water: An Efficient System for the Reduction of Aldehydes to Alcohols
Indian Journal of Chemistry, Sect. B. 33, 182-183 (1994) (

Retrieved by Azole:

For fallen_Angel:
2,4,5-trimethoxybenzaldehyde from vanillin
J. Chem. Soc. (C), 2222-2229 (1969) (

pyrylium salts by Ac2O/HClO4 diacylation of olefins
Tetrahedron Lett., 4643-4644 (1968) (

For Rhodium:

A Convenient Preparation of Conjugated Nitro Olefins by Electrochemical Method.
A. Kunai, Y. Yanagi, and K. Sasaki
Tetrahedron Lett., 24(41), 4443-4444 (1983). (

Studies on the Formation of Complex Oxidation and Condensation Products of Phenols. A Contribution to the Investigation of the Origin and Nature of Humic Acid. Part I. - Studies of the Reactivity of Simple Monocyclic Quinones. (Added 03-09-04):
H. G. H. Erdtman
Proc. Roy. Soc. London., Ser. A, 143, 177-191 (1933). (

Studies on the Formation of Complex Oxidation and Condensation Products of Phenols. Part II.
Coupling of Simple Phenols and Quinones to Diphenyl Derivatives.
(Added 03-09-04):
H. G. H. Erdtman
Proc. Roy. Soc. London., Ser. A, 143, 191-222 (1933). (

For pHarmacist:
A One-step Ester to Hydrocarbon Reduction.
Donald C. Wigfield and Kevser Taymaz
Tetrahedron Lett., 49, 4481-4484 (1973). (

Diels-Alder route to precursors of anthranilic acid derivatives
K. Gewald,
Chem. Ber., 99, 1002 (1966) (

For Chimimanie:
Indoles.  XXXII.  Synthesis of tryptophols.
Grandberg, I. I.; Moskvina, T. P.
Khimiya Geterotsiklicheskikh Soedinenii, 1972(10), 1366-7 (
This article is reviewed in the book "Preparative Chemistry of Indole" (in Russian) along with several other articles concerning tryptophols by the same author (I.I.Grandberg).

Darstellung und Reduktion von Indolyl-(3)-aminomethylketonen
K.Bodendorf, A.Walk
Arch. Pharm.  (1961),  294  484-7 (

Il Farmaco, Ed. Sc., 14, 854-866 (1959). (
Il Farmaco, Ed. Sc., 16, 483-491 (1961). (
Il Farmaco, Ed. Sc., 16, 492-501 (1961). (

For GC_MS:
A new synthesis of methoxalen.
P Nore, E Honkanen
J. Heterocycl. Chem., 17 (1980) 985-987 (

For Ruthenium:
The Reimer-Tiemann Reaction, Enhanced by Ultrasound (Added 03-15-04):
John C. Cochran and Margaret G. Melville
Synth. Commun., 1990, 20(4), 609-616.

For Nicodem:
Ethyl nitroacetate from acetoacetic ester (Added 03-15-04):
V. M. Rodionov, E. V. Machinskaya, and V. M. Belikov
Zh. Obshch. Khim., 18, 917-920 (1948) (in Russian).

For Lego:
An efficient method for the conversion of phenolic Mannich bases to C-methylated phenols. Synthesis of 3,6-dimethylcatechol. (Added 02-15-04):
Sinhababu, A. K.; Borchardt, R. T.
Synthetic Communications, 12(12), 983-988 (1982). (

Selective ring C-methylation of hydroxybenzaldehydes via their Mannich bases. (Added 02-15-04):
Sinhababu, A. K.; Borchardt, R. T.
Synthetic Communications, 13(8), 677-683 (1983). (

Alkene Reductions Employing Ethyl Acetate - Hydroxylamine, a Useful New Source of Diimide
P. A. Wade, N. V. Amin
Synthetic Communications, 12(4),  287-91 (1982). (

An improved preparation of phenylacetone.
J. Kizlink
Chemicke Listy (1990), 84(9),  993-4.

Oxidation of nitromethane by manganese(III) acetate:  novel formation of methyl radical.
Srivastava, Ranjan P.; Seth, M.; Bhaduri, A. P.
Indian Journal of Chemistry, Section B:  Organic Chemistry Including Medicinal Chemistry  (1989), 28B(1), 65-6.

Synthesis of nitroalkanes from bromoalkanes by phase-transfer catalysis.
Sane, Pramodchandra V.; Sharma, Man Mohan
Organic Preparations and Procedures International (1988), 20(6), 598-9.

Preparation of N-unsubstituted thioamides by a modified Willgerodt-Kindler reaction.
You, Qidong; Zhou, Houyuan; Wang, Qizhou; Lei, Xinghan
Organic Preparations and Procedures International (1991), 23(4), 435-8. (

Improved synthesis of phenylacetamides by the Willgerodt reaction with microwave heating.
Strauss, Christopher R.; Trainor, Robert W.
Organic Preparations and Procedures International (1995),  27(5), 552-5. (

Selective reduction of nitro compounds with titanium(II) reagents.
J. George and S. Chandrasekaran
Synthetic Communications, 13(6), 495-9 (1983). (

The following articles are in Russian:

Methylation of phenol with methyl formate.
Nasadyuk, V. A.; Fedevich, E. V.; Pazderskii, Yu. A.; Moiseev, I. I.   
Izvestiya Akademii Nauk SSSR, Seriya Khimicheskaya, 1989,  787-90. (

Reactions of hydrazine derivatives. XVII. New synthesis of α-methyltryptophol.
Grandberg, I. I.; Kost, A. N.; Terent'ev, A. P.
Zhurnal Obshchei Khimii, 27, 3342-5 (1957) (

Heating 10.8 g. PhNHNH2, 10.2 g. AcCH2CH2CH2OH, and 6 ml. AcOH 0.5 hr. at 100° gave after addn. of NH4OH and extn. with Et2O 88.5% PhNHN:CMeCH2CH2CH2OH (I), b8 194-6°, m. 60-6°.  Reaction of 51 g. AcCH2CH2CH2Cl and 48.6 g. PhNHNH2 in EtOH gave after 1 hr. on steam bath 52.4% 1-phenyl-3-methyl-1,4,5,6-tetrahydropyridazine, b6 197-8° (picrate, m. 226.5°).  Heating 15.7 g. PhNHNH2 and 15.3 g. AcCH2CH2CH2OH 1 hr. on steam bath, heating in vacuo to 150° to remove H2O, addn. of 0.2 g. Cu2Cl2 and heating to 230° 2 hrs. gave 69.4% a-methyltryptophol (II), b7-8 202-4°, m. 52-5° (picrate, m. 132°); use of ZnCl2 as catalyst gave 63% yield.  I and AcCl in dioxane-CCl4 gave 33.4% O-acetyl-a-methyltryptophol, b3-4 196-204° (picrate, m. 131.5°), also formed from II and Ac2O at reflux.  II and PBr3 in Et2O gave after an aq. treatment 70.3% a-methyl-b-(b-bromoethyl)indole, m. 58°, which with aq. Me2NH at 100° gave 66.5% a-methyl-b-(b-dimethylaminoethyl)indole, b21 204-5°, m. 93-5° (picrate, m. 176°).  Cf. Hoshinyo, et al. C.A. 29, 79757.

For 1kplateau:
Supramolecular catalytic systems based on cyclodextrins in Wacker oxidation. (Added 03-09-04):
E. A. Karakhanov, A. Ya. Zhuchkova, T. Yu. Filippova, A. L. Maximov
Neftekhimiya, 43(4), 302-307 (2003) (

   The article is written in Russian. There exists an English version of the journal (the page number you cited probably refers to the translation) but I've never seen it. Most of the references are in English. The yields are not very encouraging, and the modified cyclodextrins applied are not commercially available. Anyway, I'll try to translate the article if you like.

Wacker oxidation of various 1-alkenes (1-hexene to 1-dodecene) and p-substituted styrenes was performed under 5 MPa pressure of O2 in a biphasic system water - alkene in the presence of palladium sulfate and modified beta-cyclodextrins (see Fig. 1). Copper salts were applied as a co-catalyst. Oxidation of 1-alkenes led to the corresponding methyl ketones; styrenes gave mixtures of acetophenones and arylacetaldehydes.

Retrieved by Zamboni:

For Chimimanie:
a-Asarone congeners as hypolipidemic agents. Pseudoreceptor versus minireceptor modeling. (Added 03-09-04):   
Filipek, Slawomir; Lozowicka, Bozena.    Department of Chemistry,  Warsaw University,  Warsaw,  Pol.   
Acta Poloniae Pharmaceutica  (2000),  57(Suppl.),  106-109. (

Indigo to alpha-Methyltryptamine (Added 03-09-04):
S. Pietra and G. Tacconi
Farmaco, Ed. Sci 13, 893 (1958) (
(If anyone wants to see the 1957 Farmaco article that's listed as a reference in the 1958 Farmaco article, I have that, too. Of course there is a US patent which describes the process: Patent US3282959)

For Rhodium:
The part that I copied before my money ran out for the xerox machine:
5-Hydroxyvanillin to Myristicinaldehyde in 77% Yield (Added 03-09-04):
Taniguchi, Eiji; Imamura, Keiichi; Ishabashi, Fumito; Matsui, Toshio; Nishio, Akira
Agric. Biol. Chem.; 53(3) 631-644 (1989) (

Isomerization of some allylbenzenes in a microwave batch reactor (Added 03-09-04):
Le, Ngoc Thach; Strauss, Christopher R.
Tap Chi Hoa Hoc 38(1), 76-79 (2000) (

For Kinetic:
Zinc chloride catalysed 2,2-dialkyl benzodioxole acylations with acetic anhydride, yields over 90% (Added 03-09-04):
Indian J.Chem.Sect.B; 38; 2; 1999; 137 - 140. (

Retrieved by pHarmacist:

For Chimimanie:
Analogs of amphetamine. 6. 2,5-Dimethoxy-4-methyl- and 2,5-dimethoxy-alpha,4-dimethylphenylalanines
Beng T. Ho, L. Wayne Tansey, Jen-Tzaw Huang;
J. Med. Chem.; 1971; 14(11); 1132-1133 (

Roger M. Pinder, Keith Brewster;
J. Med. Chem.; 1971; 14(7); 650-651 (

Dihydroxynitrobenzaldehydes and hydroxymethoxynitrobenzaldehydes: synthesis and biological activity as catechol-O-methyltransferase inhibitors
Rosa A. Perez, Eldiberto Fernandez-Alvarez, Ofelia Nieto, F. Javier Piedrafita;
J. Med. Chem.; 1992; 35(24); 4584-4588 (

Phenylalkylamines with potential psychotherapeutic utility. 1. 2-Amino-1-(2,5-dimethoxy-4-methylphenyl)butane
Robert T. Standridge, Henry G. Howell, Jonas A. Gylys, Richard A. Partyka, Alexander T. Shulgin;
J. Med. Chem.; 1976; 19(12); 1400-1404 (

beta-Chloroethylamines related to mescaline
Cooper, Paul D.
Journal of Medicinal Chemistry 16, 1057-9 (1973) (

Retrieved by Lugh:

For Lego:
New Sulfur Derivatives Of Indoles
Rocz. Chem.; 50; 1976; 603. (
Lego's voice: N,N-substituted indol-3-yl-thioacetamides could bee valuable precursors for N,N-substituted tryptamines as thioamides are easily reduced to the corresponding amines.

For Potter:
Acetophenone to Phenylacetone: PhCOCH3 + CH2N2 --AlCl3--> P2P (50%)
Katalysierte Homologisierung Cycloaliphatischer und Aliphatischer Ketone mit Diazoalkanen
Eugen Müller, Martin Bauer
Ann. Chem. 654, 92-111 (1962) (

For Barium:
The Darzen Condensation, Part I
J. Chem. Soc. C (1970), 1154 (

The Darzen Condensation, Part III
J. Chem. Soc., Perkin Trans. 2 (1975), 805 (

Stereochemical Control of the Darzens Condensation
J.Chem. Soc., Chem. Commun. (1977), 902 (

Synthesis of Glycidic esters in a two-phase solid-liquid system
Synth. Commun. (1982), 12, 355 (

For pHarmacist:
Indolylalkylamines From Arylhydrazines and gamma- and delta-Halocarbonyl Compounds (Review)
Grandberg, I. I.
Chem. Heterocycl. Compd. (engl. Transl.) 1974, 10, 501. (

Structural Correlation between Apomorphine and LSD:
Involvement of Dopamine as well as Serotonin in the Actions of Hallucinogen

Dave E. Nichols
J. Theor. Biol. 59, 167-177 (1976) (

For Rhodium:
Sodium borohydride: A versatile reagent in the reductive N-monoalkylation of -amino acids and -amino methyl esters
Can. J. Chem./Rev. Can. Chim. 80(7): 779-788 (2002) (

Benzene Hydrocarbons with a Pseudo Allyl Side Chain: Methovinylbenzene and its Homologues. Study of Certain Molecular Migrations. Second Part. Study of Molecular Transpositions which Accompany the Transformation of -Glycols and their Derivatives into Aldehydes and Ketones.
Tiffeneau, M.
Ann. chim. phys., [8], Vol 10, pp 322-78 (1908) (
Abstract: Post 446645 (Rhodium: "Glycols, halohydrins & epoxides to P2P", Novel Discourse)

Preparation of Optically Active -aminopropiophenones by asymmetric transformation
H. Takamatsu
J. Pharm. Soc. Japan, Vol. 76, 1219-1222 (1956) (

Trifluoroacetylation of Methylated-Derivatives of Tryptamine and Serotonine by Different Reagents: Synthesis, Spectroscopic Characterizations, and Separations by Capillary-Gas-Chromatography
Haefelinger, Guenter; Nimtz, Manfred; Horstmann, Volker; Benz, Thomas
Zeitschrift für Naturforschung B, Vol 54, No 3, 397-414 (1999) (

For GC_MS:
Sodium Percarbonate: A Mild Reagent for Conversion of Tosylhydrazones and Nitroalkanes to Carbonyl Compounds
C Narayana, NK Reddy. GW Kabalka
Synth. Commun. 22(17), 2587-2592 (1992) (

For Chimimanie:
Synthesis and some properties of 1,2-dihydro-4,7-dihydroxycyclobuta{b}naphthalene-3,8-dione and 1,2,5,6-tetrahydro-4,7-dihydroxydicyclobuta{b,g}naphthalene-3,8-dione.
Watabe, Takashi; Oda, Masaji
Chemistry Letters (10), 1791-4 (1984) (

Comparison of stimulants and hallucinogens on shuttle avoidance in rats
Davis, W. M.; Hatoum, H. T.
General Pharmacology 18(2), 123-8 (1987) (

Synthesis and turnover of 3H-5-hydroxytryptamine in the lateral cerebroventricle
Kantak, K. M.; Wayner, M. J.; Tilson, H. A.; Dwoskin, L. P.; Stein, J. M.
Pharmacology, Biochemistry and Behavior 8(2), 153-61 (1978) (

Evaluation of substituted-amphetamine hallucinogens using the cat limb flick model
Rusterholz, D. B.; Spratt, J. L.; Long, J. P.; Barfknecht, C. F.
Communications in Psychopharmacology  1(6), 589-92 (1977) (

Further studies on BL-3912A:  effects on avoidance behavior of rats with low baselines and on reaction thresholds to electric footshock
Tilson, Hugh A.; Chamberlain, John H.; Gylys, Jonas A.
Pharmacology, Biochemistry and Behavior 6(6),  627-30 (1977) (

For Potter:
Peyote Alkaloids IX: Identification and Synthesis of 3-Demethylmescaline, a Plausible Intermediate in the Biosynthesis of the Cactus Alcaloids
G,J, Kapadia, Y. N. Vaishnav, M. B. E. Fayez
J. Pharm. Sci. 58(9), 1157-1159 (1969) (

For Sonson:
The stereoisomers of 4-Methylaminorex
R. F. Klein, A.R. Sperling, D. A. Cooper, T. C. Kram
Journal of Forensic Sciences 34(4), 962-979 (1989) (
____ ___ __ _

For Rhodium:

J. Anal. Toxicol. 24(7), 602-5 (2000)

Tetrahedron Letters 24(41), 4443-4444 (1983)

M.Lefler, R.Adams. J.Am.Chem.Soc. 59, 2252 (1937) (Added 02-15-04):

and the English translation of Zh.Org.Khim. 19(11), 2288-2294 (1983):
J.Org.Chem.USSR (Engl.Transl.) 1997-2002 (1983) (Added 02-15-04):

The formation and chemical properties of diastereomeric 1,2-Dimethyl-3-phenylaziridine (Added 02-15-04):
T. Taguchi & M. Kojima
Chem. Pharm. Bull. 7, 103-107 (1959)

The Synthesis of 14C-diethylamine and lysergic acid diethylamide (Added 02-15-04):
Journal of Labelled Compounds and Radiopharmaceuticals 10:(2), 207 (1974)

A Study of the Precursors, Intermediates and Reaction By-Products on the Synthesis of MDMA and its Application to Forensic Drug Analysis. (Added 02-15-04):
Renton, R.J., Cowie, J.S. and Oon, M.C.
Forensic Science International 60, 189-202 (1993)

Synthesis of (R)- and (S)-amphetamine-d3 from the corresponding phenylalanines
Gal J.
J. Labelled Comp. Radiopharm. 13, 3-9 (1977)

For moo:
Preparation of nitroethane. latest addition (03-19-04):
Desseigne, Gerard; Giral, Henri.
Memorial des Poudres, 34, 49-53 (1952).

For Lego:
Plant Physiol. 42: 520-524

For Chimimanie:
Arzneimittel-Forschung  (2001),  51(7),  535-544

Identification of new secondary metabolites of methoxyphenamine in man., (Added 02-15-04):
McKay, G.; Cooper, J. K.; Hawes, E. M.; Roy, S. D.; Midha, K. K.
Xenobiotica  (1983),  13(4),  257-64.

Phytochemistry (Elsevier)  (1981),  20(5),  1164-5

Chemical & Pharmaceutical Bulletin  (1980),  28(10),  2948-59

For pHarmacist:
Chem. Pharm. Bull., 1985, 33, 3696

For Vitus_Verdegast:
Aromatic Chlorination by Aqueous Sodium Hypochlorite (Added 03-09-04):
C.Y. Hopkins and M. J. Chisholm
Can. J. Research B, 24, 208 (1946)

For josef_k:
Synthesis of Ketomebidone Precursors via Phase-Transfer Catalysis (Added 03-09-04):
T. Cammack & P. C. Reeves
Can. J. Research B, 24, 208 (1946)

For Antoncho:
Sites of action of gamma-hydroxybutyrate (GHB)--a neuroactive drug with abuse potential. (Added 03-09-04):
Tunnicliff G.
Journal of toxicology. Clinical toxicology. 35(6), 581-90 (1997)

Request by Psychokitty:

Isomerization of pseudoephedrine into ephedrine...
Izv. Akad. Nauk Kaz. SSR, Ser. Tekhn. i Khim. Nauk 1963 (3), 20-7 (pub. 1964) (Russ); cf Tr. Inst. Khim. Nauk, akad. Nauk Kaz. SSR 4, 127-34 (1959).

Retrieved by Flogiston, addendum by Polythenesam/Rhodium:

Reference retrieved and can be read at Post 425116 (Flogiston: "Изомеризация псевдоэфедрина в эфедрин.", Russian HyperLab)

Edit: "Chem. Abs. Vol 2, 3348 has something about isomerizing ephedrine and pseudoephedrine into the other isomer (in equilibrium) using HCl." /PolytheneSam 
That CA article has been scanned and can be read at /Rhodium

Retrieved by Herr_Ovalmeister:
Here's Russian patent SU 239341 in TIFF format.

Phenyl-2-Propanal isomerization to P2P:

Hydro- and solvatolytic and intramolecular oxidation-reduction. II. Acid and acid-salt catalysis in the isomerisation of aldehydes to ketones.
S. N. Danilov
Zhurnal Obshchei Khimii, 18(11), 2000-2007 (1948). (

Post 424552 (Dionket: "J Org Chem USSR ?", Russian HyperLab)
Post 446720 (Timmy: "So it is...", Russian HyperLab)
Post 476441 (azole: "as requested by java", Russian HyperLab)

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Date: 10-01-23, Release: 1.6 (10-04-15), Links: static, unique